TGFβRI-IN-1
目录号: A18800
TGFβRI kinase 抑制剂
TGFβRI-IN-1 是一种口服活性且选择性的 TGFβ 受体类型 I (TGFβRI) 激酶抑制剂,其 IC50 值分别针对 TGFβRI 和 TGFβRII 为 2 nM 和 7.6 μM。
Discription | TGFβRI-IN-1 is an oral active and selective TGFβ receptor type I (TGFβRI) kinase inhibitor, with IC50 values of 2 nM and 7.6 μM for TGFβRI and TGFβRII, respectively. |
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目录号 | A18800 |
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分子式 | C20H14D3N5O2 |
分子量 | 362.4 |
CAS号 | 1950628-94-0 |
SMILES | CC(NC1=NC=CC(C(N2)=C(C3=NC=C(OC([2H])([2H])[2H])C=C3)C4=C2C=CC=N4)=C1)=O |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2