TGR5-Receptor-Agonist
目录号: A13732
TGR5(GPCR19) 激动剂
TGR5 受体激动剂是一种强效的 TGR5(GPCR19) 激动剂,在 U2-OS 细胞测试中显示出提高的效力(pEC50 = 6.8),以及在黑色素细胞中也表现出较高的效力(pEC50 = 7.5)。
Discription | TGR5 Receptor Agonist is a potent TGR5(GPCR19) agonist, showed improved potency in the U2-OS cell assay (pEC50 = 6.8) and in melanophore cells (pEC50 = 7.5). |
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目录号 | A13732 |
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分子式 | C18H14Cl2N2O2 |
分子量 | 361.22 |
CAS号 | 1197300-24-5 |
SMILES | CC1=C(C(=NO1)C2=CC=CC=C2Cl)C(=O)N(C)C3=CC=C(C=C3)Cl |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2