Tipifarnib (Zarnestra)

目录号: A10935

FTase inhibitor

Tipifarnib (Zarnestra)

Tipifarnib (Zarnestra) Chemical Structure

CAS NO. 192185-72-1

Tipifarnib (Zarnestra) is a farnesyltransferase inhibitor that inhibits the Ras kinase in a post translational modification step before the kinase pathway becomes hyperactive.

库存: 现货

规格 价格 数量
5 mg
¥ 1,500.00
10 mg
¥ 2,500.00
25 mg
¥ 4,500.00
100 mg
¥ 8,000.00
10mM * 1mL in DMSO
¥ 2,060.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

Tipifarnib (Zarnestra) is a farnesyltransferase inhibitor that inhibits the Ras kinase in a post translational modification step before the kinase pathway becomes hyperactive.
Targets
FTase
0.6 nM
In vitro (25°C) DMSO 14 mg/mL (28.6 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 15% Captisol/citrate vehicle 5 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.43 mL 102.17 mL 204.33 mL
0.5 mM 4.09 mL 20.43 mL 40.87 mL
1 mM 2.04 mL 10.22 mL 20.43 mL
5 mM 0.41 mL 2.04 mL 4.09 mL

*The above data is based on the productmolecular weight 489.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A10935
MECHANISM OF ACTION Inhibitor
M. Wt 489.4
Formula C27H22Cl2N4O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 192185-72-1
Synonyms IND 58359, R115777
SMILES CN1C=NC=C1[C@@](C2=CC=C(C=C2)Cl)(C3=CC4=C(C=C3)N(C(=O)C=C4C5=CC(=CC=C5)Cl)C)N

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