Tonapofylline

目录号: A21328

adenosine A1 receptor antagonist

Tonapofylline

Tonapofylline Chemical Structure

CAS NO. 340021-17-2

Tonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure.

库存: 现货

规格 价格 数量
5 mg
¥ 2,250.00
10 mg
¥ 3,880.00
50 mg
¥ 11,500.00
100 mg
¥ 23,000.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

Tonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.01 mL 120.05 mL 240.09 mL
0.5 mM 4.8 mL 24.01 mL 48.02 mL
1 mM 2.4 mL 12 mL 24.01 mL
5 mM 0.48 mL 2.4 mL 4.8 mL

*The above data is based on the productmolecular weight 416.51. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A21328
作用机制 Antagonist (拮抗剂)
M. Wt 416.51
Formula C22H32N4O4
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 340021-17-2
Synonyms BG 9928
SMILES O=C(O)CCC1(CC2)CCC2(C(N3)=NC(N(CCC)C(N4CCC)=O)=C3C4=O)CC1

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