UNC-1999

目录号: A13166

EZH2/EZH1 Inhibitor

UNC-1999

UNC-1999 Chemical Structure

CAS NO. 1431612-23-5

UNC1999 is the first orally bioavailable inhibitor that has high in vitro potency for wildtype and mutant EZH2 as well as EZH1.

库存: 现货

规格 价格 数量
5 mg
¥ 600.00
10 mg
¥ 1,100.00
25 mg
¥ 2,200.00
50 mg
¥ 3,500.00
10mM * 1mL in DMSO
¥ 1,270.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

UNC1999 is the first orally bioavailable inhibitor that has high in vitro potency for wildtype and mutant EZH2 as well as EZH1.
Targets
EZH2 (Cell-free assay) EZH1 (Cell-free assay)
2 nM45 nM
In vitro DMSO 100 mg/mL (175.51 mM)
Water <1 mg/mL (<1 mM)
Ethanol 100 mg/mL (175.51 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.55 mL 87.76 mL 175.52 mL
0.5 mM 3.51 mL 17.55 mL 35.1 mL
1 mM 1.76 mL 8.78 mL 17.55 mL
5 mM 0.35 mL 1.76 mL 3.51 mL

*The above data is based on the productmolecular weight 569.74. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

目录号 A13166
MECHANISM OF ACTION Inhibitor
M. Wt 569.74
Formula C33H43N7O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1431612-23-5
Synonyms UNC 1999, UNC1999
SMILES CCCC1=C(C(=O)NC(=C1)C)CNC(=O)C2=C3C=NN(C3=CC(=C2)C4=CN=C(C=C4)N5CCN(CC5)C(C)C)C(C)C

产品标签

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。

Product Questions

Product Questions

No Questions
Keywords:购买 UNC-1999 | UNC-1999 供应商 | 订购 UNC-1999 | UNC-1999 价格 | UNC-1999 生产商 | 订单 UNC-1999 | UNC-1999 代理商 | 购买 1431612-23-5| 1431612-23-5 供应商 | 订购 1431612-23-5 | 1431612-23-5 价格 | 1431612-23-5 生产商 | 订单 1431612-23-5 | 1431612-23-5 代理商|buy UNC-1999 | UNC-1999 Supplier | purchase UNC-1999 | UNC-1999 cost | UNC-1999 manufacturer | order UNC-1999 | UNC-1999 distributor | buy 1431612-23-5| 1431612-23-5 Supplier | purchase 1431612-23-5 | 1431612-23-5 cost | 1431612-23-5 manufacturer | order 1431612-23-5 | 1431612-23-5 distributor
Rewards