UNC0379 TFA
目录号: A22036
SETD8 抑制剂
UNC0379 TFA 是一种选择性的、与底物竞争的赖氨酸甲基转移酶 SETD8 (KMT5A) 抑制剂,其 IC50 为 7.3 μM;相较于其他 15 种甲基转移酶具有选择性。
Discription | UNC0379 TFA is a selective, substrate-competitive inhibitor of lysine methyltransferase SETD8 (KMT5A) with an IC50 of 7.3 μM; selective over 15 other methyltransferases. |
---|
目录号 | A22036 |
---|---|
分子式 | C25H36F3N5O4 |
分子量 | 527.58 |
CAS号 | 1620401-83-3 |
SMILES | COC1=C(OC)C=C2C(N=C(N3CCCC3)N=C2NCCCCCN4CCCC4)=C1.O=C(O)C(F)(F)F |
其他名称 | UNC 0379, UNC-0379 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2