UNC0379
目录号: A14320
SETD8 HMTase 抑制剂
UNC0379 是一种选择性的、与底物竞争的赖氨酸甲基转移酶 SETD8 的抑制剂。其对 SETD8 的亲和力通过 ITC（等温滴定量热法）和 SPR（表面等离子体共振）研究得到确认。
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生物活性
| Discription | UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8. Its affinity to SETD8 was confirmed by ITC (isothermal titration calorimetry) and SPR (surface plasmon resonance) studies. | ||
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产品信息
| 目录号 | A14320 |
|---|---|
| 分子式 | C23H35N5O2 |
| 分子量 | 413.28 |
| CAS号 | 1620401-82-2 |
| SMILES | COC1=C(C=C2C(=C1)C(=NC(=N2)N3CCCC3)NCCCCCN4CCCC4)OC |
| 其他名称 | UNC-0379, UNC 0379 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | 79 mg/mL (191.02 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 24.2 mL | 120.98 mL | 241.97 mL |
| 0.5 mM | 4.84 mL | 24.2 mL | 48.39 mL |
| 1 mM | 2.42 mL | 12.1 mL | 24.2 mL |
| 5 mM | 0.48 mL | 2.42 mL | 4.84 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 1620401-82-2 | 1620401-82-2 供应商 | 1620401-82-2 花费 | 1620401-82-2 生产商 | 订购 1620401-82-2 | 1620401-82-2 代理商