UNC0379

目录号: A14320

SETD8 HMTase inhibitor

UNC0379 Chemical Structure

CAS NO. 1620401-82-2

UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8. Its affinity to SETD8 was confirmed by ITC (isothermal titration calorimetry) and SPR (surface plasmon resonance) studies.

库存: 现货

规格 价格 数量
5 mg
¥ 800.00
10 mg
¥ 1,350.00
25 mg
¥ 2,800.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8. Its affinity to SETD8 was confirmed by ITC (isothermal titration calorimetry) and SPR (surface plasmon resonance) studies.
靶点信息
SETD8
7.9 μM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.2 mL 120.98 mL 241.97 mL
0.5 mM 4.84 mL 24.2 mL 48.39 mL
1 mM 2.42 mL 12.1 mL 24.2 mL
5 mM 0.48 mL 2.42 mL 4.84 mL

*The above data is based on the productmolecular weight 413.28. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A14320
MECHANISM OF ACTION Inhibitor
M. Wt 413.28
Formula C23H35N5O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1620401-82-2
Synonyms UNC-0379, UNC 0379
SMILES COC1=C(C=C2C(=C1)C(=NC(=N2)N3CCCC3)NCCCCCN4CCCC4)OC

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