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Vasopressin antagonist 1867

Vasopressin antagonist 1867

Name: Vasopressin antagonist 1867
SKU: A16188

目录号: A16188

V1b receptor 拮抗剂

Vasopressin antagonist 1867 Chemical Structure

CAS NO. 909391-88-4

Vasopressin antagonist 1867，可口服和选择性V1b受体拮抗剂（hV1b抑制作用的IC50值为3 nM，相对于hV1a，hV2和hOT表现出> 1000倍的选择性）。

库存：现货

规格	价格	数量
5 mg	￥ 1,200.00
10 mg	￥ 2,000.00
50 mg	￥ 8,000.00

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生物活性

Vasopressin antagonist 1867，可口服和选择性V1b受体拮抗剂（hV1b抑制作用的IC50值为3 nM，相对于hV1a，hV2和hOT表现出> 1000倍的选择性）。

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	20.3 mL	101.5 mL	203 mL
0.5 mM	4.06 mL	20.3 mL	40.6 mL
1 mM	2.03 mL	10.15 mL	20.3 mL
5 mM	0.41 mL	2.03 mL	4.06 mL

*The above data is based on the productmolecular weight 492.61. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A16188
作用机制	Antagonist (拮抗剂)
M. Wt	492.61
Formula	C28H36N4O4
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	909391-88-4
Synonyms	Compound 12i
SMILES	CC(C)NC(=O)CN1C(=NC2=C(C1=O)C=C(C=C2)OCCCN3CCCCC3)C4=CC(=CC=C4)OC