VLX1570
目录号: A16853
DUB 抑制剂
VLX1570 是蛋白酶体 DUB 活性的竞争性抑制剂,在体外的 IC50 约为 10 μM。
Discription | VLX1570 is a competitive inhibitor of proteasome DUB activity, with an IC50 of ~10?μM in vitro. | |||||
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Cell Research |
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目录号 | A16853 |
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分子式 | C23H17F2N3O6 |
分子量 | 469.39 |
CAS号 | 1431280-51-1 |
SMILES | O=C1/C(CN(C(C=C)=O)CC/C1=C/C2=CC=C(F)C([N+]([O-])=O)=C2)=C\C3=CC=C(F)C([N+]([O-])=O)=C3 |
其他名称 | VLX 1570, VLX-1570 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 79 mg/mL (168.3 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 21.3 mL | 106.52 mL | 213.04 mL |
0.5 mM | 4.26 mL | 21.3 mL | 42.61 mL |
1 mM | 2.13 mL | 10.65 mL | 21.3 mL |
5 mM | 0.43 mL | 2.13 mL | 4.26 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2