Zibotentan (ZD4054)

目录号: A11006

ETA-receptor Antagonist

Zibotentan (ZD4054) Chemical Structure

CAS NO. 186497-07-4

Zibotentan (ZD4054)is an orally administered, potent and specific ETA-receptor (endothelin A receptor) antagonist (IC50 = 21 nM).

库存: 现货

规格 价格 数量
5 mg
¥ 900.00
10 mg
¥ 1,600.00
50 mg
¥ 4,500.00
100 mg
¥ 7,500.00
10mM * 1mL in DMSO
¥ 1,350.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

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Zibotentan (ZD4054)is an orally administered, potent and specific ETA-receptor (endothelin A receptor) antagonist (IC50 = 21 nM).
靶点信息
ET-A
21 nM
In vitro (25°C) DMSO 24 mg/mL (56.54 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.56 mL 117.81 mL 235.63 mL
0.5 mM 4.71 mL 23.56 mL 47.13 mL
1 mM 2.36 mL 11.78 mL 23.56 mL
5 mM 0.47 mL 2.36 mL 4.71 mL

*The above data is based on the productmolecular weight 424.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11006
MECHANISM OF ACTION Antagonist
M. Wt 424.4
Formula C19H16N6O4S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 186497-07-4
Synonyms ZD-4054
SMILES CC1=CN=C(C(=N1)OC)NS(=O)(=O)C2=C(N=CC=C2)C3=CC=C(C=C3)C4=NN=CO4

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