Carbonic Anhydrase

Catalog No.Inhibitor Name Carbonic AnhydraseCarbonic Anhydrase ICarbonic Anhydrase IICarbonic Anhydrase IVCarbonic Anhydrase IXCarbonic Anhydrase XII
A10333Dorzolamide HCl
*
****
***
A14959U-104
*
*
**
****
A11673Tioxolone
**
A11765Brinzolamide
****
***
A10303Dichlorphenamide
A15859Acetazolamide
***
A13594Benzenesulfonamide

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

12 个项目

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  1. Ethoxzolamide

    Catalog No. A17359
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    Carbonic anhydrase inhibitor
    Ethoxzolamide is a carbonic anhydrase inhibitor with Ki of 1 nM. 了解更多
  2. Dorzolamide HCL

    Catalog No. A10333
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    carbonic anhydrase 抑制剂
    Dorzolamide HCl是一种碳酸酐酶抑制剂。它是一种抗青光眼剂,以滴眼剂的形式局部使用。盐酸度尔佐胺用于降低开角型青光眼和高眼压患者的眼内压升高。 了解更多
  3. Tioxolone

    Catalog No. A11673
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    Carbonic anhydrase 抑制剂
    Tioxolone是一种抗痤疮制剂。 了解更多
  4. Brinzolamide

    Catalog No. A11765
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    Carbonic anhydrase 抑制剂
    Brinzolamide是一种碳酸酐酶抑制剂,IC50为3.19 nM。 了解更多
  5. Diclofenamide

    Catalog No. A10303
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    Carbonic anhydrase 抑制剂
    Diclofenamide (or dichlorphenamide)是一种磺酰胺和间二氨磺酰苯类的碳酸酐酶抑制剂。 了解更多
  6. Indisulam (E7070)

    Catalog No. A12325
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    Carbonic anhydrase inhbitor
    Indisulam (E7070)是一种碳酸酐酶抑制剂,也是一种靶向细胞周期G1期的新型合成磺酰胺。 了解更多
  7. Punicalagin

    Catalog No. A12105
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    Carbonic anhydrase 抑制剂
    Punicalagin是一种鞣花单宁,一种酚类化合物。它是一种高活性碳酸酐酶抑制剂。 了解更多
  8. Punicalin

    Catalog No. A12106
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    Carbonic anhydrase 抑制剂
    Punicalin是一种高活性碳酸酐酶抑制剂。 了解更多
  9. DTP348

    Catalog No. A14410
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    CAIX 抑制剂/ radiosensitizer
    DTP348是双重CAIX抑制剂/放射增敏剂。 了解更多
  10. U-104

    Catalog No. A14959
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    Carbonic anhydrase (CA) 抑制剂
    U-104是碳酸酐酶IX(CAIX)的新型脲基磺酰胺抑制剂。 了解更多
  11. Acetazolamide

    Catalog No. A15859
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    Carbonic Anhydrase 抑制剂
    Acetazolamide是一种有效的碳酸酐酶(CA)抑制剂,在临床实践中通常用作迅速降低眼内压(IOP)的直接且容易获得的选择。 了解更多
  12. Benzenesulfonamide

    Catalog No. A13594
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    Carbonic anhydrase 抑制剂
    Benzenesulfonamide是碳酸酐酶的抑制剂。 了解更多

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