|HER1/EGFR (Cell-free assay)|
|In vitro (25°C)||DMSO||3 mg/mL (6.97 mM)|
|Water||<1 mg/mL (<1 mM)|
|Ethanol||<1 mg/mL (<1 mM)|
|In vivo||1% DMSO, 0.5% CMC Na and 15% Captisol||20 mg/mL|
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|0.1 mM||23.26 mL||116.31 mL||232.61 mL|
|0.5 mM||4.65 mL||23.26 mL||46.52 mL|
|1 mM||2.33 mL||11.63 mL||23.26 mL|
|5 mM||0.47 mL||2.33 mL||4.65 mL|
*The above data is based on the productmolecular weight 429.9 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|MECHANISM OF ACTION||Inhibitor|
|Storage||at -20°C 3 years Powder|
|Synonyms||CP-358774, OSI-774, NSC 718781|
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