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￥ 0.00 5-HT Receptors
16 个项目
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Flopropione
Catalog No. A16550 5-HT1A receptor antagonist/COMT inhibitorFlopropione是5-HT1A受体拮抗剂，也是儿茶酚-邻甲基转移酶（COMT）抑制剂。 了解更多 -
Vortioxetine
Catalog No. A21266 5-HT1A/5-HT1B/5-HT3A/5-HT7 receptor/SERT inhibitorVortioxetine is a inhibitor of 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT, with Ki values of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively. 了解更多 -
Vilazodone D8
Catalog No. A21876 SSR inhibitor / 5-HT1A receptor partial agonistVilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多 -
Eplivanserin mixture
Catalog No. A21987 serotonin reuptake inhibitor/5-HT2A receptor antagonistEplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多 -
Vilazodone
Catalog No. A11116 Serotonin reuptake 抑制剂Vilazodone充当5-羟色胺再摄取抑制剂（IC50 = 0.5 nM）和5-HT1A受体部分激动剂（IC50 = 0.2 nM； IA =?60-70％）。 了解更多 -
Sibutramine hydrochloride
Catalog No. A12397 -
Levomilnacipran HCl
Catalog No. A14391 -
Edivoxetine HCl
Catalog No. A13865 -
Norfluoxetine
Catalog No. A13458 serotonin uptake 抑制剂Norfluoxetine是抗抑郁药氟西汀的活性代谢物，抑制5-羟色胺的摄取，pKi值为7.35.1氟西汀的S-对映体的5-羟色胺再摄取阻断能力是R-对映体的20倍（pKis分别为7.86和6.51）。 了解更多 -
Atomoxetine HCl
Catalog No. A13424 norepinephrine (NE) transporter 抑制剂Atomoxetine HCl是SLC6A2的一种竞争性特异性抑制剂，同时在大鼠下丘脑突触体中显示出微弱的ST和DAT抑制作用。 了解更多 -
Asenapine HCl
Catalog No. A15002 adrenergic receptor/5-HT receptor 抑制剂Asenapine hydrochloride抑制肾上腺素能受体（α1，α2A，α2B，α2C）的Ki为0.25-1.2 nM，还抑制5-HT受体（1A，1B，2A，2B，2C，5A，6、7），Ki为0.03- 4.0 nM。 了解更多 -
Desvenlafaxine succinate hydrate
Catalog No. A15491 serotonin (5-HT)/norepinephrine (NE) reuptake 抑制剂Desvenlafaxine succinate hydrate是一种新型5-羟色胺(5-HT)转运蛋白 和去甲肾上腺素(NE)转运蛋白重吸收抑制剂，Ki值分别为40.2 nM和558.4 nM 了解更多 -
Eucalyptol
Catalog No. A15662 -
Nefazodone hydrochloride
Catalog No. A17622 5-HT2 receptors inhibitorNefazodone HCl is an inhibitor of 5-HT2 receptors, SERT, NET, and hERG K+ channels used to treat mood disorders. It decreases immobility time in the forced swim test. 了解更多
16 个项目
每页