CGRP Receptor

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  1. CGRP 8-37 (human)

    Catalog No. A16949
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    CGRP receptor 拮抗剂
    CGRP 8-37 (human)是人降钙素基因相关肽(hCGRP)片段,也是CGRP受体的拮抗剂。序列:Val-Thr-His-Arg-Leu-Ala-Gly-Leu-Leu-Ser-Arg-Ser-Gly-Gly-Val-Val-Lys-Asn-Asn-Phe-Val-Pro-Thr-Asn- Val-Gly-Ser-Lys-Ala-Phe;VTHRLAGLLSRSGGVVKNNFVPTNVGSKAF。 了解更多
  2. Olcegepant

    Catalog No. A11512
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    CGRP1 receptor
    Olcegepant is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. 了解更多
  3. Ubrogepant

    Catalog No. A21670
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    CGRP antagonist
    Ubrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine. 了解更多
  4. Olcegepant hydrochloride

    Catalog No. A21900
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    CGRP1 receptor antagonist
    Olcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP. 了解更多
  5. MK 3207 HCl

    Catalog No. A10598
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    CGRP Receptor 拮抗剂
    MK 3207 hydrochloride是一种有效的CGRP受体拮抗剂,IC50为0.12 nM。 了解更多
  6. MK-0974 (Telcagepant)

    Catalog No. A11255
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    CGRP receptor 拮抗剂
    MK-0974 (Telcagepant)是人和恒河猴CGRP受体的有效和选择性拮抗剂。 了解更多
  7. BMS-927711

    Catalog No. A13102
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    CGRP receptor 拮抗剂
    BMS-927711是一种有效的,选择性的,竞争性的人降钙素基因相关肽(CGRP)受体拮抗剂,已显示出体内功效,而没有血管收缩作用。 了解更多
  8. MK-3207

    Catalog No. A15165
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    CGRP Receptor 拮抗剂
    MK-3207是一种有效且口服可生物利用的CGRP受体拮抗剂(IC50 = 0.12 nM;Ki = 0.024 nM);对人类AM1,AM2,CTR和AMY3具有高度选择性。 了解更多

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