HDAC

Catalog No.Inhibitor Name HDAC HDAC1 HDAC2 HDAC3 HDAC4HDAC5 HDAC6 HDAC7 HDAC8 HDAC9 HDAC10 HDAC11 HD1 HD2
A10979Vorinostat
****
A10611Entinostat
**
*
A10518Panobinostat
****
A10947Trichostatin A
****
A10586Mocetinostat
**
**
*
*
A10122Belinostat
***
A11920Romidepsin
***
***
A10560MC1568
*
A11042Tubastatin A HCl
*
***
A10488Givinostat
****
****
A10516Dacinostat
***
A10246CUDC-101
****
****
***
****
***
***
****
**
**
**
***
A10830Pracinostat
***
**
***
***
***
*
**
**
**
***
**
A11152PCI-34051
*
*
****
*
A10337Droxinostat
*
*
*
A10700Abexinostat
****
***
****
***
**
***
A13218RGFP966
**
A11037AR-42
***
A11940Ricolinostat
**
***
***
*
*
****
*
**
A11964Tacedinaline
*
*
*
**
A11153CUDC-907
****
****
****
**
*
***
**
**
****
****
A11355M344
**
A10954Tubacin
****
A13139RG2833
***
****
A12556Resminostat
***
***
**
A15489BRD73954
*
***
**
A11361BG45
*
*
**
A143544SC-202
*
*
*
A16431CAY10603
**
****
A14341LMK-235
***
****
A14032Nexturastat A
****
A14128TMP269
**
**
***
***
A14197HPOB
*
*
*
***
*
*
A12722Scriptaid
A12616Tasquinimod
A11042Tubastatin A
***

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. PCI-24781 (Abexinostat)

    Catalog No. A10700
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    HDAC 抑制剂
    PCI-24781 (Abexinostat)是一种广谱苯基异羟肟酸HDAC抑制剂。 了解更多
  2. Scriptaid

    Catalog No. A12722
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    HDAC 抑制剂
    Scriptaid是一种HDAC抑制剂(组蛋白脱乙酰基酶)。 了解更多
  3. Vorinostat (SAHA)

    Catalog No. A10979
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    HDAC 抑制剂
    Vorinostat (SAHA)是HDAC的抑制剂,抑制脱乙酰和导致双方超乙酰化组蛋白和转录因子的积累。 了解更多
  4. LAQ824 (NVP-LAQ824, Dacinostat)

    Catalog No. A10516
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    HDAC 抑制剂
    LAQ824 (NVP-LAQ824)是一种有效的新型组蛋白去乙酰化酶抑制剂,具有显著的抗多发性骨髓瘤活性。 了解更多
  5. NCH 51

    Catalog No. A15355
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    HDAC 抑制剂
    NCH 51是细胞可渗透的前药,可在细胞内转化为有效的HDAC抑制剂,IC50为48 nM。 了解更多
  6. Belinostat (PXD101)

    Catalog No. A10122
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    HDAC 抑制剂
    Belinostat(PXD101)是一种HDAC抑制剂,可抑制HeLa细胞提取物中的HDAC活性,IC50为27 nM。 了解更多
  7. SB939 ( Pracinostat )

    Catalog No. A10830
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    HDAC 抑制剂
    SB939 (Pracinostat)是HDAC的口服抑制剂,对I,II和IV类HDAC具有选择性,在体外HDAC1活性测定中显示IC50值为77 nM。 了解更多
  8. AR-42 (HDAC-42)

    Catalog No. A11037
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    HDAC 抑制剂
    AR-42 (HDAC-42)是一种新型的HDAC抑制剂,通过下调本构激活的Kit表现出对恶性肥大细胞系的生物学活性。 了解更多
  9. Apicidin

    Catalog No. A12745
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    HDAC 抑制剂
    Apicidin是一种有效的组蛋白脱乙酰基酶(HDAC)抑制剂,具有潜在的抗癌活性。 了解更多
  10. NSC 3852

    Catalog No. A15356
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    HDAC 抑制剂
    NSC 3852是HDAC(组蛋白脱乙酰基酶)抑制剂。 了解更多
  11. CUDC-101

    Catalog No. A10246
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    HDAC 抑制剂
    CUDC-101是一种抑制多种靶标的新型化合物,旨在抑制HDAC,EGFR和Her2。 了解更多
  12. JNJ-26481585 (Quisinostat)

    Catalog No. A10492
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    HDAC 抑制剂
    JNJ-26481585 (Quisinostat)是一种pan-HDAC抑制剂,对HDAC1具有显著的效力(IC(50),0.16 nmol/L)。 了解更多
  13. Valproic acid

    Catalog No. A17323
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    HDAC inhibitor
    Valproic acid is an HDAC inhibitor, with IC50 in the range of 0.5 and 2 mM, also inhibits HDAC1 (IC50, 400 μM), and induces proteasomal degradation of HDAC2; Valproic acid sodium salt is used in the treatment of epilepsy, bipolar disorder and prevention of migraine headaches. 了解更多
  14. Splitomicin

    Catalog No. A14221
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    NAD(+)-dependent histone deacetylase Sir2p 抑制剂
    Splitomicin是一种选择性的NAD(+)-依赖性组蛋白脱乙酰基酶Sir2p抑制剂,IC50为60 uM,在基于细胞的测定中显示出更高的活性。 了解更多
  15. HDAC inhibitor

    Catalog No. A13405
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    HDAC 抑制剂
  16. Ac-Lys-AMC

    Catalog No. A18461
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    fluorescent substrate for HDAC
    Ac-Lys-AMC (Hexanamide), also termed MAL, is a fluorescent substrate for histone deacetylase HDACs. 了解更多
  17. ST7612AA1

    Catalog No. A14418
    HDAC 抑制剂
    ST7612AA1是新型的有效HDAC抑制剂,具有潜在的抗癌活性。 了解更多
  18. R306465

    Catalog No. A15437
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    HDAC 抑制剂
    R306465是一种新型的基于异羟肟酸酯的组蛋白脱乙酰基酶(HDAC)抑制剂,在临床前模型中具有针对实体和血液恶性肿瘤的广谱抗肿瘤活性。 了解更多
  19. M344

    Catalog No. A11355
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    HDAC 抑制剂
    M344是HDAC的有效抑制剂,IC50为100 nM,能够诱导细胞分化。 了解更多
  20. ITSA-1

    Catalog No. A16127
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    HDAC 抑制剂
    ITSA-1具有膜渗透性,可以特异性抑制TSA对HDAC(组蛋白脱乙酰基酶)的抑制,但不能抑制其他HDAC抑制剂。 了解更多
  21. BML-210

    Catalog No. A15935
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    HDAC 抑制剂?
    BML-210是HDAC抑制剂。BML-210诱导宫颈癌细胞中的生长抑制和凋亡并调节HDAC和DAPC复合物的表达水平。 了解更多

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