Estrogen Receptors

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  1. Tamoxifen Citrate

    Catalog No. A10885
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    Estrogen receptor 拮抗剂
    Tamoxifen Citrate是哺乳动物甾醇异构酶的选择性和有效抑制剂。 了解更多
  2. Fulvestrant R enantiomer

    Catalog No. A21545
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    estrogen receptor antagonist
    Fulvestrant R enantiomer (ICI 182780 R enantiomer; ZD 9238 R enantiomer; ZM 182780 R enantiomer) is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM. 了解更多
  3. H3B-6545 Hydrochloride

    Catalog No. A21629
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    estrogen receptor covalent antagonist
    H3B-6545 Hydrochloride is an oral, selective estrogen receptor covalent antagonist (SERCA). 了解更多
  4. AZD9496 maleate

    Catalog No. A21726
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    estrogen receptor (ERα) antagonist
    AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多
  5. Enclomiphene citrate

    Catalog No. A21830
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    oestrogen receptor antagonist
    Enclomiphene citrate is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property. 了解更多
  6. Endoxifen

    Catalog No. A12639
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    Estrogen receptor 拮抗剂
    Endoxifen是他莫昔芬的次生代谢产物。它是负责他莫昔芬在ER阳性乳腺癌中有效性的主要代谢物。Endoxifen Z-isomer抑制hERG, 这种作用具有浓度依赖性, IC50值为1.6μM。 了解更多
  7. AZD9496

    Catalog No. A15822
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    estrogen receptor downregulator and 拮抗剂
    AZD9496是一种有效的生物选择性雌激素受体下调剂和拮抗剂。 了解更多
  8. (E/Z)-4-hydroxy Tamoxifen

    Catalog No. A12532
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    Estrogen receptor 拮抗剂
    (E/Z)-4-hydroxy Tamoxifen是他莫昔芬的活性代谢产物,是一种选择性雌激素受体(ER)调节剂,广泛用于乳腺癌的治疗和化学预防治疗。 了解更多
  9. H3B-6545

    Catalog No. A20100
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    Estrogen receptor antagonist
    H3B-6545 is an oral, selective estrogen receptor covalent antagonist (SERCA). 了解更多
  10. XCT 790

    Catalog No. A13299
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    ERRα 拮抗剂/inverse 激动剂
    XCT 790是ERRα的强效特异性反向激动剂。 了解更多
  11. IRL-2500

    Catalog No. A13638
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    ETBR 拮抗剂
    IRL-2500是一种有效的选择性ETBR拮抗剂。它显示了对ETB受体的一些选择性(对于ETB和ETA受体,IC50值分别为1.3和94 nM)。 了解更多

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