P-gp

Catalog No.Inhibitor Name P-gpOther
A10549Zosuquidar 3HCl
**
A11584Tariquidar
***
A12324Elacridar (GF120918)
BCRP

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. P-gp inhibitor 1

    Catalog No. A13384
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    P-gp inhibitor
    P-gp inhibitor 1 is a novel inhibitor reversing P-glycoprotein-mediated multidrug resistance. 了解更多
  2. Norverapamil hydrochloride

    Catalog No. A12249
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    P-gp inhibitor
    Norverapamil hydrochloride ((??)-Norverapamil hydrochloride), an N-demethylated metabolite of Verapamil, is a L-type calcium channel blocker and a P-glycoprotein (P-gp) function inhibitor. 了解更多
  3. TTT-28

    Catalog No. A13033
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    ABCB1 (P-gp/MDR1) inhibitor
    TTT-28 is a synthesized thiazole-valine peptidomimetic, a novel selective inhibitor of ABCB1 (P-gp/MDR1) with high efficacy and low toxicity. 了解更多
  4. Zosuquidar

    Catalog No. A15289
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    P-gp 抑制剂
    Zosuquidar是P-糖蛋白介导的多药耐药性的有效调节剂,Ki为60 nM。 了解更多
  5. Elacridar hydrochloride

    Catalog No. A15077
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    P-gp 抑制剂
    Elacridar hydrochloride是一种P-糖蛋白抑制剂,已在体内和体外用作P-糖蛋白(Pgp)的工具抑制剂,以研究转运蛋白在处理各种测试分子中的作用。 了解更多
  6. Biricodar

    Catalog No. A21464
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    P-glycoprotein/MRP-1 modulator
    Biricodar (VX-710) is a modulator of P-glycoprotein and MRP-1; shows effective chemosensitizing activity in multidrug resistant cells. 了解更多
  7. FD 12-9

    Catalog No. A18393
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    P-gp/BCRP dual 抑制剂
    FD 12-9 is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively. Anti-glioblastoma activity. 了解更多
  8. KS-176

    Catalog No. A16195
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    BCRP 抑制剂
    KS-176是乳腺癌抗性蛋白(BCRP)多药转运蛋白的有效和选择性抑制剂(在Pheo A和Hoechst 33342分析中,IC50值分别为0.59和1.39 uM)。 了解更多
  9. MC 70 HCl

    Catalog No. A16080
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    P-gp 抑制剂
    MC 70 HCl是有效的P-gp抑制剂(EC50 = 0.69 uM)。 了解更多
  10. Biricodar dicitrate (VX-710 dicitrate)

    Catalog No. A13533
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    P-gp modulator
    Biricodar dicitrate (VX-710 dicitrate)是P-糖蛋白和MRP-1的调节剂;在多药耐药细胞中显示出有效的化学增敏活性。 了解更多
  11. Laniquidar

    Catalog No. A13532
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    P-gp 抑制剂
    Laniquidar是第三代P-gp抑制剂,已在临床试验中用于调节多药耐药转运蛋白。 了解更多
  12. ONT-093

    Catalog No. A13531
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    P-gp 抑制剂
    ONT-093是口服可生物利用的P-糖蛋白泵抑制剂,可潜在逆转接受癌症化学疗法的患者的多药耐药性。 了解更多
  13. XR9576

    Catalog No. A13961
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    P-glycoprotein 抑制剂
    XR9576是一种 P-glycoprotein (P-gp) 抑制剂,Kd值为5.1 nM。正在研究中作为抗癌多药耐药性的佐剂。 了解更多
  14. Cynarin

    Catalog No. A12004
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    Cynarin是朝鲜蓟中的一种酚类化合物。它具有抗氧化剂和胆汁特性。它是一种潜在的免疫抑制剂。 了解更多
  15. Selamectin

    Catalog No. A12363
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    Selamectin是一种局部寄生虫药和抗蠕虫药,用于狗和猫,以治疗和预防犬中的心丝虫,跳蚤,耳螨,螨和某些种类的壁虱感染,并预防心丝虫,跳蚤,耳螨,钩虫和round虫 在猫中。 了解更多
  16. Tariquidar (XR9576)

    Catalog No. A11584
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    P-gp 抑制剂
    Tariquidar (XR9576)是一种P-糖蛋白药物外排泵抑制剂。 了解更多
  17. Elacridar (GF120918)

    Catalog No. A12324
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    P-gp & BCRP 抑制剂
    Elacridar (GF120918)是一种原型BCRP抑制剂,可抑制Bcrp1介导的转运。 了解更多
  18. PSC-833 (Valspodar)

    Catalog No. A11080
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    MDR1/P-gp 抑制剂
    PSC-833 (Valspodar)是一种P-糖蛋白(P-gp)调节剂,可抑制P-gp介导的多药耐药性(MDR)。 了解更多
  19. LY335979 (Zosuquidar 3HCl)

    Catalog No. A10549
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    P-gp modulator
    LY335979 (Zosuquidar trihydrochloride)是一种强效高选择性P-gp抑制剂。 了解更多

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