AChE

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  1. (±)-Huperzine A

    Catalog No. A21003
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    AChE inhibitor
    (??)-Huperzine A, an active Lycopodium alkaloid extracted from traditional Chinese herb, is a potent, selective and reversible acetylcholinesterase (AChE) inhibitor and has been widely used in China for the treatment of Alzheimer's disease (AD). 了解更多
  2. (+)-Phenserine

    Catalog No. A20993
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    cholinesterase noncompetitive inhibitor
    (+)-Phenserine is a novel selective cholinesterase noncompetitive inhibitor with an IC50 of 45.3 μM. 了解更多
  3. (R)-Rivastigmine D6 tartrate

    Catalog No. A21454
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    cholinesterase inhibitor
    (R)-Rivastigmine D6 (tartrate) is the deuterium labeled (R)-Rivastigmine, which is an cholinesterase inhibitor. 了解更多
  4. Acetyllovastatin

    Catalog No. A19111
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    AChE inhibitor
    Acetyllovastatin, a acetate of Lovastatin, presentes a moderate inhibitory effect against the enzyme acetylcholinesterase with an IC50 of 79 μg/mL. Lovastatin has been found to display antifungal activity, and suppresses proliferation of a number of transformed cell lines. 了解更多
  5. MHP 133

    Catalog No. A20058
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    AChE /M1/M2/5HT4/I2 inhibitor
    MHP 133 is a drug with multiple CNS targets, and inhibits acetylcholinesterase (AChE) with Ki of 69 μM; also active against muscarinic M1 and M2 receptors, serotonin 5HT4 receptors, and imidazole I2 receptors. 了解更多
  6. Galanthamine

    Catalog No. A12483
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    AChE inhibitor
    Galanthamine is a potent acetylcholinesterase (AChE) inhibitor with an IC50 of 500 nM. 了解更多
  7. Edrophonium chloride

    Catalog No. A17794
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    acetylcholinesterase inhibitor
    Edrophonium Chloride, also known as Tensilon, is an acetylcholinesterase inhibitor used in cardiac arrhythmias and in the diagnosis of myasthenia gravis. Edrophonium Chloride has also been used as an antidote to curare principles. 了解更多
  8. Nerolidol

    Catalog No. A17599
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    AChE inhibitor
    Nerolidol is a synthetic AChE inhibitor and F0F1-ATP synthase modulator. It acts as a sedative, inhibits growth of bacteria and fungi, and decreases the mitochondrial transmembrane electric potential to induce cell death in hepatocarcinoma cells. 了解更多
  9. Pralidoxime Iodide

    Catalog No. A17526
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    Cholinesterase Reactivator
    Pralidoxime iodide is a Cholinesterase Reactivator. 了解更多
  10. Tacrine HCl

    Catalog No. A17374
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    AChE & butyrylcholinesterase inhibitor
    Tacrine is a derivative of aminoacridine that functions as an inhibitor of both acetylcholinesterase (AChE) and butyrylcholinesterase (IC50s = 31 and 26.5 nM, respectively). 了解更多
  11. Pitofenone Hydrochloride

    Catalog No. A17053
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    Antispasmodic Agent
    Pitofenone Hydrochloride是抗痉化合物。它是乙酰胆碱酯酶活性的有效抑制剂。 了解更多
  12. Tacrine HCl Hydrate

    Catalog No. A16970
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    AChE and BChE 抑制剂
    Tacrine hydrochloride hydrate是乙酰(AChE)和丁酰胆碱酯酶(BChE)的抑制剂,IC50分别为31 nM和25.6 nM。 了解更多
  13. Rivastigmine

    Catalog No. A14096
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    AChE and BChE 抑制剂
    Rivastigmine是一种胆碱酯酶抑制剂(IC50 = 5.5 uM),可同时抑制丁酰胆碱酯酶和乙酰胆碱酯酶。 了解更多
  14. Pulegone

    Catalog No. A14353
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    AChE 抑制剂
    Pulegone是在许多精油中发现的单萜化合物。 了解更多
  15. Acotiamide hydrochloride trihydrate

    Catalog No. A15782
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    AChE 抑制剂
    Acotiamide hydrochloride trihydrate是一种在日本获准用于治疗餐后饱胀,上腹胀气和功能性消化不良引起的早饱的药物。 了解更多
  16. Deoxyvasicine HCl

    Catalog No. A13925
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    AChE 抑制剂
    Desoxypeganine hydrochloride是一种AChE(乙酰胆碱酯酶)抑制剂,已用于治疗阿尔茨海默氏痴呆症。 了解更多
  17. Donepezil

    Catalog No. A13079
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    AChE 抑制剂
    Donepezil是一种非竞争性乙酰胆碱酯酶抑制剂,可以很容易地穿过血脑屏障并增加皮质乙酰胆碱的浓度。众所周知,多奈哌齐是研究阿尔茨海默病的有用工具。 了解更多
  18. Neostigmine bromide (Prostigmin)

    Catalog No. A10635
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    AChE 抑制剂
    Neostigmine bromide是一种可逆的乙酰胆碱酯酶抑制剂,可与AChE的阴离子结合位点结合。 了解更多
  19. Donepezil hydrochloride

    Catalog No. A10330
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    cholinesterase 抑制剂
    Donepezil hydrochloride是一种中枢可逆的乙酰胆碱酯酶抑制剂。 了解更多
  20. Rivastigmine tartrate

    Catalog No. A11719
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    AChE 抑制剂
    Rivastigmine tartrate是一种双重胆碱酯酶抑制剂(ChEI)。它同时抑制丁酰胆碱酯酶(BChE)和乙酰胆碱酯酶(AChE)。 了解更多
  21. Galanthamine hydrobromide

    Catalog No. A10416
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    AChE 抑制剂
    Galanthamine hydrobromide是一种乙酰胆碱酯酶抑制剂,IC50为14 nM。 了解更多

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