HDAC

Catalog No.Inhibitor Name HDAC HDAC1 HDAC2 HDAC3 HDAC4HDAC5 HDAC6 HDAC7 HDAC8 HDAC9 HDAC10 HDAC11 HD1 HD2
A10979Vorinostat
****
A10611Entinostat
**
*
A10518Panobinostat
****
A10947Trichostatin A
****
A10586Mocetinostat
**
**
*
*
A10122Belinostat
***
A11920Romidepsin
***
***
A10560MC1568
*
A11042Tubastatin A HCl
*
***
A10488Givinostat
****
****
A10516Dacinostat
***
A10246CUDC-101
****
****
***
****
***
***
****
**
**
**
***
A10830Pracinostat
***
**
***
***
***
*
**
**
**
***
**
A11152PCI-34051
*
*
****
*
A10337Droxinostat
*
*
*
A10700Abexinostat
****
***
****
***
**
***
A13218RGFP966
**
A11037AR-42
***
A11940Ricolinostat
**
***
***
*
*
****
*
**
A11964Tacedinaline
*
*
*
**
A11153CUDC-907
****
****
****
**
*
***
**
**
****
****
A11355M344
**
A10954Tubacin
****
A13139RG2833
***
****
A12556Resminostat
***
***
**
A15489BRD73954
*
***
**
A11361BG45
*
*
**
A143544SC-202
*
*
*
A16431CAY10603
**
****
A14341LMK-235
***
****
A14032Nexturastat A
****
A14128TMP269
**
**
***
***
A14197HPOB
*
*
*
***
*
*
A12722Scriptaid
A12616Tasquinimod
A11042Tubastatin A
***

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. MGCD0103 (Mocetinostat)

    Catalog No. A10586
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    HDAC 抑制剂
    MGCD0103 (Mocetinostat)是一种苯甲酰胺组蛋白脱乙酰基酶抑制剂,主要抑制组蛋白脱乙酰基酶1(HDAC1),但也抑制HDAC2,HDAC3和HDAC11。 了解更多
  2. CI994 (Tacedinaline)

    Catalog No. A11964
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    HDAC 抑制剂
    CI994 (Tacedinaline)是一种组蛋白脱乙酰基酶(HDAC)抑制剂,可在活细胞中诱导组蛋白超乙酰化。 了解更多
  3. Resminostat hydrochloride

    Catalog No. A15220
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    HDAC 抑制剂
    Resminostat hydrochloride是HDAC1/3/6的有效抑制剂(IC50 = 43-72 nM);对HDAC8的效力较低,IC50为877 nM。 了解更多
  4. HDAC-IN-7

    Catalog No. A21252
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    HDAC1/2/3/10 inhibitor
    HDAC-IN-7 (Chidamide impurity) is an impurity of Chidamide. Chidamide is a potent and orally bioavailable HDAC enzymes class I (HDAC1/2/3) and class IIb (HDAC10) inhibitor. 了解更多
  5. Trichostatin-A (TSA)

    Catalog No. A10947
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    HDAC 抑制剂
    Trichostatin-A (TSA)是抑制HDAC 1、3、4、6和10,IC50值约为20 nM。 了解更多
  6. CUDC-907 (Fimepinostat)

    Catalog No. A11153
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    PI3K/HDAC 抑制剂
    CUDC-907 (Fimepinostat)是针对PI3K和HDAC的单一小分子抑制剂,作用于PI3Kα和HDAC1/2/3/10,IC50分别为19 nM和1.7 nM/5 nM/1.8 nM/2.8 nM。 了解更多
  7. RG2833 (RGFP109)

    Catalog No. A13139
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    HDAC 抑制剂
    RG2833 (RGFP109)是一种脑渗透性HDAC抑制剂,IC50为60 nM,HDAC1和HDAC3为50 nM。 了解更多
  8. PCI-24781 (Abexinostat)

    Catalog No. A10700
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    HDAC 抑制剂
    PCI-24781 (Abexinostat)是一种广谱苯基异羟肟酸HDAC抑制剂。 了解更多
  9. Romidepsin (FK228 ,Depsipeptide)

    Catalog No. A11920
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    HDAC 抑制剂
    Romidepsin (FK228,Depsipeptide)抑制HDAC1和HDAC2,IC50分别为1.6 nM和3.9 nM,但相对较弱地分别抑制HDAC4和HDAC6,IC50值为25 nM和79 nM。 了解更多
  10. KD 5170

    Catalog No. A15354
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    HDAC 抑制剂
    KD 5170是一种新型的基于巯基酮的组蛋白脱乙酰基酶抑制剂,在体外和体内均表现出广谱的抗肿瘤活性。 了解更多
  11. LBH589 (Panobinostat)

    Catalog No. A10518
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    HDAC 抑制剂
    LBH589是异羟肟酸,用作非选择性HDAC抑制剂,HDAC1的IC5o为0.23 nM。 了解更多
  12. Parthenolide ((-)-Parthenolide)

    Catalog No. A10698
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    Parthenolide ((-)-Parthenolide), Nuclear Factor-κB抑制剂,可特异性地耗尽HDAC1蛋白,而不影响其他I/II类 HDACs。促进MDM2的泛素化并激活p53的细胞功能。 了解更多
  13. MS-275 (Entinostat)

    Catalog No. A10611
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    HDAC 抑制剂
    MS-275 (Entinostat)是一种有效的HDAC抑制剂,对HDAC1和HDAC3的IC50分别为0.3和8uM。 了解更多
  14. Pyroxamide (NSC 696085)

    Catalog No. A10764
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    HDAC 抑制剂
    Pyroxamide (NSC 696085)是亲和纯化的HDAC1的有效抑制剂,可导致乙酰化核心组蛋白在用该试剂培养的MEL细胞中积累。 了解更多
  15. Resminostat

    Catalog No. A12556
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    HDAC 抑制剂
    Resminostat,也称为RAS2410,是一种有效的I和II类组蛋白脱乙酰基酶(HDAC)抑制剂。它结合并抑制HDAC,从而导致高度乙酰化的组蛋白的积累。选择性的抑制HDAC1/3/6,IC50为42.5 nM/50.1 nM/71.8 nM,作用于HDAC8效果弱,IC50为877 nM。 了解更多
  16. Valproic acid

    Catalog No. A17323
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    HDAC inhibitor
    Valproic acid is an HDAC inhibitor, with IC50 in the range of 0.5 and 2 mM, also inhibits HDAC1 (IC50, 400 μM), and induces proteasomal degradation of HDAC2; Valproic acid sodium salt is used in the treatment of epilepsy, bipolar disorder and prevention of migraine headaches. 了解更多
  17. SR-4370

    Catalog No. A16899
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    HDAC 抑制剂
    SR-4370是HDAC抑制剂。SR-4370对HDAC1,HDAC2和HDAC3的IC50值分别为0.5 uM,0.1 uM和0.06 uM。 了解更多
  18. UF010

    Catalog No. A15781
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    HADC 抑制剂
    UF010是一种有效的选择性HADC抑制剂,对于HDAC 3、2、1和8分别具有IC50?0.06 uM,0.1 uM,0.5 uM和1.5 uM。它的选择性是其他HDAC的6倍以上。 了解更多
  19. CM-675

    Catalog No. A18741
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    PDE5/HDAC-1 inhibitor
    CM-675 is a dual phosphodiesterase 5 (PDE5) and class I histone deacetylases-selective inhibitor, with IC50 values of 114 nM and 673 nM for PDE5 and HDAC1, respectively. CM-675 has potential to treat Alzheimer??s disease. 了解更多
  20. Tinostamustine (EDO-S101)

    Catalog No. A18342
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    HDAC inhibitor
    EDO-S101 is a pan HDAC inhibitor; inhibits HDAC1, HDAC2 and HDAC3 with IC50 values of 9, 9 and 25 nM, respectively. 了解更多
  21. Domatinostat (4SC-202)

    Catalog No. A14354
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    HDAC 抑制剂
    4SC-202是生物利用的苯甲酰胺和人I类组蛋白脱乙酰基酶(HDACs)同工酶1、2和3的抑制剂,具有潜在的抗肿瘤活性。 了解更多
  22. BRD-6929

    Catalog No. A12511
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    HDAC1/HDAC2 inhibitor
    BRD-6929 (Cpd-60) is a brain-penetrant, selective inhibitor of HDAC1 and HDAC2 (IC50=?1 and 8 nM), extracted from patent US2018360927. 了解更多
  23. BG45

    Catalog No. A11361
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    HDAC 抑制剂
    BG45是一种HDAC I类抑制剂,对HDAC3具有选择性(IC50 = 289 nM)。它抑制HDAC1,HDAC2和HDAC6的效力大大降低(IC50分别为2、2和> 20μM)。 了解更多
  24. TC-H 106

    Catalog No. A15357
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    HDAC 抑制剂
    TC-H 106是一种慢速,紧密结合的I类HDAC(组蛋白脱乙酰基酶)抑制剂。 了解更多

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