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￥ 0.00 Factor Xa
| Catalog No. | Inhibitor Name | Factor Xa | Other |
|---|---|---|---|
| A10800 | Rivaroxaban | ** | Prothrombinase |
| A10082 | Apixaban | **** | |
| A14317 | Edoxaban | *** | Thrombin,FIXa |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
17 个项目
每页
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BMS-654457
Catalog No. A21704 Factor XIa (FXIa) inhibitorBMS-654457 is a small-molecule, reversible inhibitor of factor XIa (FXIa), binding with human and rabbit FXIa with Kis of 0.2 and 0.42 nM, respectively. 了解更多 -
RWJ-445167
Catalog No. A12154 dual inhibitor of thrombin and factor XaRWJ-445167 (3DP-10017) is a dual inhibitor of thrombin and factor Xa with Ki of 4.0 nM and 230 nM, respectively, exhibiting potent antithrombotic activity. 了解更多 -
Fondaparinux Sodium
Catalog No. A17918 factor Xa inhibitorFondaparinux sodium is a factor Xa inhibitor to form the high affinity binding site for the anti-coagulant factor antithrombin III (ATIII). 了解更多 -
Edoxaban tosylate
Catalog No. A15076 -
5-R-Rivaroxaban
Catalog No. A14979 Factor Xa 抑制剂5-R-Rivaroxaban是利伐沙班的（R）对映异构体。利伐沙班是一种新型的口服直接Xa因子抑制剂，在晚期开发中用于预防和治疗血栓栓塞性疾病。 了解更多 -
Edoxaban (tosylate Monohydrate)
Catalog No. A14317 Factor Xa 抑制剂Edoxaban (tosylate Monohydrate)是选择性Factor Xa抑制剂，Ki为0.561 nM。 了解更多 -
Betrixaban
Catalog No. A12518 FXa 抑制剂Betrixaban是一种抗凝血药，可作为直接Xa因子抑制剂。它具有强大的，口服活性和对因子Xa的高度选择性，由于其低hERG亲和力而从一组相似的化合物中选择。 了解更多 -
Letaxaban (TAK-442)
Catalog No. A12871 factor Xa 抑制剂Letaxaban (TAK-442)是一种有效的，选择性的，口服活性的Xa抑制剂，是一种四氢嘧啶-2（1H）-衍生物。TAK-442在贫血小板的人[半最大抑制浓度（IC（50））：53 nM，TAK-442]和大鼠（IC（50）：32 nM，TAK-442）血浆中抑制内源性FXa活性。 了解更多 -
Otamixaban (FXV 673)
Catalog No. A11517 -
Rivaroxaban (Xarelto)
Catalog No. A10800 Factor Xa 抑制剂Rivaroxaban (Xarelto)是一种Factor Xa的直接抑制剂，无细胞试验中Ki和IC50分别为0.4 nM和0.7 nM。 了解更多 -
BMS-740808
Catalog No. A10158 -
Apixaban (BMS-562247-01)
Catalog No. A10082 Factor Xa 抑制剂Apixaban (BMS-562247-01)是一种抗凝剂，用于预防静脉血栓栓塞和静脉血栓栓塞事件。 了解更多
17 个项目
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