PAK

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  1. IPA-3

    Catalog No. A21182
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    PAK1 inhibitor
    IPA-3 is a selective non-ATP competitive PAK1 inhibitor with IC50 of 2.5 μM, and shows no inhibition to group II PAKs (PAKs 4-6). 了解更多
  2. GNE 2861

    Catalog No. A21697
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    PAK inhibitor
    GNE 2861 is a PAK inhibitor that displays group II selectivity. GNE 2861 inhibits PAK4, PAK5 and PAK6 with IC50s of 7.5, 36, 126 nM, respectively. 了解更多
  3. PF-3758309

    Catalog No. A11930
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    PAK4 抑制剂
    PF-3758309是抑制致癌信号和肿瘤生长的小分子p21活化激酶抑制剂。 了解更多
  4. LOR-253

    Catalog No. A13838
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    MTF-1 抑制剂
    LOR-253是人类金属调节转录因子1(MTF-1)的小分子抑制剂。 了解更多
  5. FRAX486

    Catalog No. A13691
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    PAK 抑制剂
    FRAX486是一种小分子PAK抑制剂。 了解更多
  6. KPT-9274

    Catalog No. A15506
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    PAK4 抑制剂
    KPT-9274是有口服活性的PAK4/烟酰胺磷酸核糖基转移酶 (Nampt) 抑制剂,IC50值分别为小于 100 和 125 nM。 了解更多
  7. FRAX597

    Catalog No. A12553
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    PAK 抑制剂
    FRAX597是一种小分子吡啶并嘧啶酮,是I类PAK(PAK1 IC50 = 8 nM,PAK2 IC50 = 13 nM,PAK3 IC50 = 19 nM)的有效和ATP竞争性抑制剂。 了解更多
  8. FRAX1036

    Catalog No. A16557
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    PAK inhibitor
    FRAX1036 is a PAK inhibitor with Kis of 23.3 nM, 72.4 nM, and 2.4 μM for PAK1, PAK2 and PAK4, respectively. 了解更多
  9. NVS-PAK1-1

    Catalog No. A12708
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    allosteric PAK1 inhibitor
    NVS-PAK1-1 is a potent and selective allosteric PAK1 inhibitor with an IC50 of 5 nM. 了解更多

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