RNA/DNA Polymerase

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  1. Dehydroaltenusin

    Catalog No. A21804
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    eukaryotic DNA polymerase α inhibitor
    Dehydroaltenusin is a small molecule selective inhibitor of eukaryotic DNA polymerase α, a type of antibiotic produced by a fungus with an IC50 value of 0.68 μM. 了解更多
  2. Rifabutin

    Catalog No. A10790
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    RNA polymerase 抑制剂
    Rifabutin是一种主要用于治疗肺结核的杀菌抗生素。它的作用是基于阻断细菌的DNA依赖性RNA聚合酶。 了解更多
  3. Rifampin

    Catalog No. A10791
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    RNA polymerase 抑制剂
    Rifampin是DNA依赖性的RNA聚合酶抑制剂,孕烷X受体(PXR)的原型激活剂。 了解更多
  4. T-705 (Favipiravir)

    Catalog No. A11590
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    viral RNA polymerase 抑制剂
    T-705 (Favipiravir)是一种有效的选择性RNA-dependent RNA polymerase抑制剂,在体外和体内均表现出有效的抗流感病毒活性。 了解更多
  5. Actinomycin D

    Catalog No. A13239
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    Actinomycin D是从小链霉菌中分离出来的一种代谢产物,与DNA的GpC步骤结合。抑制 DNA 修复,IC50 为 0.42 μM。该化合物可作为抗生素,并且比革兰氏阴性细菌更有效地抵抗革兰氏阳性细菌。 了解更多
  6. dmDNA31

    Catalog No. A18469
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    DNA-dependent RNA polymerase 抑制剂
    dmDNA31 is a rifamycin-class antibiotic that inhibits bacterial DNA-dependent RNA polymerase with potent bactericidal activity against S. aureus. 了解更多
  7. ddATP

    Catalog No. A18898
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    DNA polymerase 抑制剂
    dATP is a dideoxynucleotide, acts as a chain-elongating inhibitor of DNA polymerase, used for Sanger method for DNA sequencing. 了解更多
  8. DNA31

    Catalog No. A18466
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    RNA polymerase 抑制剂
    DNA31 is a potent RNA polymerase inhibitor. 了解更多
  9. Pseudouridimycin

    Catalog No. A18520
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    RNA polymerase 抑制剂
    Pseudouridimycin (PUM), an antibiotic, is a selective bacterial RNA polymerase (RNAP) inhibitor. Pseudouridimycin is a C-nucleoside analogue that is effective against both Gram-negative and Gram-positive bacteria. 了解更多
  10. ACX-362E

    Catalog No. A18560
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    DNA polymerase IIIC 抑制剂
    ACX-362E is an orally available DNA polymerase IIIC (pol IIIC) inhibitor, acts as an antimicrobial agent to treat Gram-positive infections, with a MIC50 of 2 μg/mL for C. difficile. ACX-362E displays very potent in vitro and in vivo activities against broad spectrum of C. difficile pathogens. 了解更多
  11. Triptolide (PG490)

    Catalog No. A11596
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    Triptolide (PG490)是从中草药雷公藤提取的,一种免疫抑制剂。 了解更多
  12. Thiolutin

    Catalog No. A15386
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    RNA polymerase 抑制剂
    Thiolutin是一种RNA聚合酶抑制剂,是链霉菌属细菌产生的一种基于硫的微生物抗生素。 了解更多
  13. Mithramycin A

    Catalog No. A15385
    DNA/RNA polymerase 抑制剂
    Mithramycin A是一种抗生素DNA/RNA聚合酶和可与DNA结合的转录抑制剂,可促进TNF-α的表达。Fas-配体诱导细胞凋亡。 了解更多
  14. Oncrasin 1

    Catalog No. A15333
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    RNA polymerase II 抑制剂
    Oncrasin 1是一种促凋亡物质。诱导PKC1的异常核聚集并抑制。 了解更多
  15. Valaciclovir

    Catalog No. A15270
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    DNA polymerase 抑制剂
    Valaciclovir是一种抗病毒药,用于治疗单纯疱疹,带状疱疹和B型疱疹。 了解更多
  16. BMH-21

    Catalog No. A14335
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    RNA polymerase 抑制剂
    BMH-21是有效的小分子DNA嵌入剂。BMH-21结合核糖体DNA并抑制RNA聚合酶I转录。 了解更多
  17. Delavirdine mesylate

    Catalog No. A13274
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    NNRT 抑制剂
    Delavirdine是一种有效的人类免疫缺陷病毒1型(HIV-1)逆转录酶(RT)抑制剂。 了解更多
  18. Fludarabine Phosphate (Fludara)

    Catalog No. A10395
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    Fludarabine Phosphate (Fludara)是一种用于治疗血液恶性肿瘤(血细胞癌,如白血病和淋巴瘤)的化疗药物。氟达拉滨通过干扰核糖核苷酸还原酶和dna聚合酶来抑制DNA合成。它对分裂细胞和静止细胞都有活性。 了解更多
  19. Abacavir

    Catalog No. A11115
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    Transcriptase 抑制剂
    Abacavir是一种核苷类似物逆转录酶抑制剂(NRTI);鸟苷类似物用于治疗艾滋病毒和艾滋病。 了解更多
  20. Abacavir sulfate

    Catalog No. A11120
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    Transcriptase 抑制剂
    Abacavir sulfate是一种核苷类似物逆转录酶抑制剂(NRTI)。 了解更多
  21. Tenofovir (Viread)

    Catalog No. A10908
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    HIV reverse transcriptase 抑制剂
    Tenofovir (Viread)属于一类称为核苷逆转录酶抑制剂(NRTIs)的药物。它通过减少血液中的HIV含量起作用。 了解更多

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