SGLT

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  1. Dapagliflozin (BMS512148)

    Catalog No. A10285
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    SGLT2 抑制剂
    Dapagliflozin (BMS512148)抑制钠-葡萄糖转运蛋白(SGLT2)的亚型2,后者负责肾脏中至少90%的葡萄糖重吸收。 了解更多
  2. Canagliflozin

    Catalog No. A11100
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    SGLT2 抑制剂
    canagliflozin是2型亚钠葡萄糖转运蛋白(SGLT2)的抑制剂,作用于hSGLT2,无细胞试验中IC50为2.2 nM,比作用于hSGLT1选择性高413倍。 了解更多
  3. EGT1442

    Catalog No. A10155
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    SGLT2 抑制剂
    EGT1442是有效的选择性SGLT2抑制剂。 了解更多
  4. Empagliflozin

    Catalog No. A12440
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    Empagliflozin是一种有效的选择性葡萄糖钠共转运蛋白-2抑制剂,目前正在开发中,用于治疗2型糖尿病。 了解更多
  5. LX-4211

    Catalog No. A12680
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    SGLT 抑制剂?
    LX4211是双重SGLT1/SGLT2抑制剂。 了解更多
  6. Tofogliflozin

    Catalog No. A12690
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    SGLT2 抑制剂
    Tofogliflozin是亚型2钠葡萄糖转运蛋白(SGLT2)的抑制剂,可引起肾脏中至少90%的葡萄糖重吸收。 了解更多
  7. Remogliflozin

    Catalog No. A13971
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    SGLT2 抑制剂
    Remogliflozin抑制钠葡萄糖转运蛋白(SGLT2),后者负责肾脏中的葡萄糖重吸收。 了解更多
  8. Ipragliflozin

    Catalog No. A13556
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    SGLT2 抑制剂
    Ipragliflozin是一种高效的选择性SGLT2抑制剂,IC50为2.8 nM。SGLT1/3/4/5/6的效力很小且没有效力。 了解更多
  9. Luseogliflozin

    Catalog No. A13476
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    SGLT2 抑制剂
    Luseogliflozin是由Taisho Pharmaceutical开发的一种口服活性第二代钠葡萄糖共转运蛋白2(SGLT2)抑制剂,用于治疗2型糖尿病(T2DM)患者。 了解更多
  10. T-1095

    Catalog No. A15463
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    Na+-glucose transporter 抑制剂
    T-1095是Na+-葡萄糖共转运蛋白(SGLTs)的有效和选择性抑制剂。 了解更多
  11. Canagliflozin hemihydrate

    Catalog No. A16817
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    SGLT2 抑制剂
    Canagliflozin hemihydrate是半水形式的卡格列嗪,是一种SGLT2抑制剂,在无细胞检测中hSGLT2的IC50为2.2 nM,其选择性比hSGLT1高413倍。 了解更多
  12. Ertugliflozin L-pyroglutamic acid

    Catalog No. A18054
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    SGLT inhibitor
    Ertugliflozin pidolate belongs to the class of potent and selective inhibitors of the sodium-dependent glucose cotransporters (SGLT), more specifically the type 2 which is responsible for about 90% of the glucose reabsorption from glomerulus. 了解更多
  13. SGL5213

    Catalog No. A18723
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    SGLT1 抑制剂
    SGL5213 is a potent, oral active and low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor, with IC50 values of 29 nM and 20 nM for hSGLT1 and hSGLT2, respectively. 了解更多
  14. Dapagliflozin impurity

    Catalog No. A19103
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    SGLT2 抑制剂
    Dapagliflozin impurity is an enantiomer of Dapagliflozin which is a sodium-glucose transporter 2 inhibitor. 了解更多
  15. Licogliflozin

    Catalog No. A12828
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    SGLT1/SGLT2 抑制剂
    Licogliflozin is a sodium glucose cotransporter (SGLT1 and SGLT2) inhibitor. 了解更多

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