Membrane Transporters/Ion Channels

12 个项目

每页

设置升序顺序
  1. (S)-(-)-Bay-K-8644

    Catalog No. A21164
    Quick View
    L-type Ca2+ channel agonist
    (S)-(-)-Bay-K-8644 is an agonist of L-type Ca2+ channel. (S)-(-)-Bay-K-8644 activates Ba2+ currents (IBa) (EC50=32 nM). 了解更多
  2. GV-58

    Catalog No. A21966
    Quick View
    N- and P/Q-type Ca2+ channels agonist
    GV-58 is a potent, selective N- and P/Q-type Ca2+ channels agonist with EC50 of 7.21/8.81 uM for N-type/P-Q-type Ca2+ channel; 20-fold less potent CDK inhibitor activity. 了解更多
  3. Ca2+ channel agonist 1

    Catalog No. A12186
    Quick View
    Ca2+ channel agonist/CDK2 inhibitor
    Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2, with EC50s of 14.23 μM and 3.34 μM, respectively, and is used as a potential treatment for motor nerve terminal dysfunction. 了解更多
  4. (S)-(-)-5-Fluorowillardiine

    Catalog No. A21337
    Quick View
    AMPAR agonist
    (S)-(-)-5-Fluorowillardiine is a potent and specific AMPAR agonist. 了解更多
  5. (S)-Willardiine

    Catalog No. A21957
    Quick View
    AMPA/kainate receptors agonist
    (S)-Willardiine is a potent agonist of AMPA/kainate receptors with EC50 of 44.8 uM. 了解更多
  6. D-3263

    Catalog No. A20935
    Quick View
    TRPM8 agonist
    D-3263 is an agonist of transient receptor potential melastatin member 8 (TRPM8) with potential antineoplastic activity. 了解更多
  7. Evodiamine (Isoevodiamine)

    Catalog No. A10376
    Quick View
    TRP 激动剂
    Evodiamine (Isoevodiamine)是从Tetradium植物家族中提取的一种化学物质。 它主要起产热和刺激作用。 了解更多
  8. PF-4840154

    Catalog No. A13996
    Quick View
    TrpA1 channel 激动剂
    PF-4840154是TrpA1通道的非亲电参考激动剂。基于TRPA1敲除小鼠在某些临床前发展模型中显示出几乎完全减轻了疼痛行为的事实,因此认为TRPA1通道是有吸引力的疼痛靶标。 了解更多
  9. WS 3

    Catalog No. A17047
    Quick View
    TRPM8 激动剂
    WS 3是TRPM8受体激动剂(EC50 = 3.7 μM)和凉爽剂。 了解更多
  10. WS 12

    Catalog No. A17046
    Quick View
    TRPM8 激动剂
    WS-12是有效的TRPM8激动剂,可作为凉爽剂(EC50 = 193 nM)。 了解更多
  11. Resiniferatoxin

    Catalog No. A14003
    vanilloid receptor 激动剂
    Resiniferatoxin是从大戟属(Euphorbia)属的一些植物中分离出的辣椒素的天然类似物(货号92350),包括E. resinifera。 了解更多
  12. (Z)-Capsaicin

    Catalog No. A18179
    Quick View
    TRPV1 agonist
    Zucapsaicin, also known as cis-Capsaicin, is a medication used to treat osteoarthritis of the knee and other neuropathic pain. It is applied three times daily for a maximum of three months. It reduces pain, and improves articular functions. 了解更多

12 个项目

每页

设置升序顺序
Rewards