Calcium Channels

47 个项目

每页

设置升序顺序
  1. GV-58

    Catalog No. A21966
    Quick View
    N- and P/Q-type Ca2+ channels agonist
    GV-58 is a potent, selective N- and P/Q-type Ca2+ channels agonist with EC50 of 7.21/8.81 uM for N-type/P-Q-type Ca2+ channel; 20-fold less potent CDK inhibitor activity. 了解更多
  2. JTV-519 free base

    Catalog No. A21846
    Quick View
    Ca2+-dependent blocker
    TV-519 free base (K201 free base) is a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and a partial agonist of ryanodine receptors in striated muscle. Antiarrhythmic and cardioprotective properties. 了解更多
  3. TTA-Q6(isomer)

    Catalog No. A21724
    Quick View
    T-type Ca2+ channel antagonist
    TTA-Q6(isomer) is an isomer of TTA-Q6. TTA-Q6 is a selective T-type Ca2+ channel antagonist. 了解更多
  4. TTA-Q6

    Catalog No. A21360
    Quick View
    T-type Ca2+ channel antagonist
    TTA-Q6 is a selective T-type Ca2+ channel antagonist, used in the neurological disease. 了解更多
  5. (S)-(-)-Bay-K-8644

    Catalog No. A21164
    Quick View
    L-type Ca2+ channel agonist
    (S)-(-)-Bay-K-8644 is an agonist of L-type Ca2+ channel. (S)-(-)-Bay-K-8644 activates Ba2+ currents (IBa) (EC50=32 nM). 了解更多
  6. ABT-639 hydrochloride

    Catalog No. A12571
    Quick View
    T-type Ca2+ channel blocker
    ABT-639 hydrochloride is a novel, peripherally acting, selective T-type Ca2+ channel blocker. 了解更多
  7. Caldaret

    Catalog No. A13148
    Quick View
    intracellular Ca2+ handling modulator
    Caldaret is an intracellular Ca2+ handling modulator that acts through reverse mode Na+/Ca2+ exchanger inhibition. 了解更多
  8. (S)-Amlodipine

    Catalog No. A14935
    Quick View
    Calcium channel blocker
    (S)-Amlodipine是氨氯地平的(S)-对映体,具有活性的二氢吡啶钙通道阻滞剂主要存在于(-)-异构体中。 了解更多
  9. NNC 55-0396

    Catalog No. A15188
    Quick View
    Calcium channel blocker
    NNC 55-0396是Mibefradil衍生物,是一种高度选择性的T型钙通道阻滞剂;分别在INS-1细胞中抑制Cav3.1 T型通道和HVA电流的IC50值为6.8和> 100μM。 了解更多
  10. NP118809

    Catalog No. A15192
    Quick View
    N-type calcium channel blocker
    NP118809是有效的N型钙通道阻滞剂(IC50 = 0.11 uM);对L型钙通道的选择性好。 了解更多
  11. NS6180

    Catalog No. A12405
    Quick View
    K(Ca) 3.1 channel blocker
    NS6180是一种新型有效的选择性KCa3.1通道抑制剂(IC50 = 9 nM),可防止T细胞活化和炎症反应。 了解更多
  12. Bay K 8644

    Catalog No. A15875
    Quick View
    Calcium Channel Activator
    Bay K 8644是一种有效的L型Ca2+通道选择性激活剂,IC50为17.3 nM。 了解更多
  13. Mibefradil dihydrochloride

    Catalog No. A12482
    Quick View
    Calcium channel blocker
    Mibefradil dihydrochloride是钙通道阻滞剂,对T型Ca2+通道具有中等选择性,对T型和L型通道的IC50值分别为2.7 uM和18.6 uM。 了解更多
  14. Dantrolene sodium Hemiheptahydrate

    Catalog No. A16146
    Quick View
    Dantrolene sodium是一种骨骼肌松弛剂,其通过干扰肌肉纤维中的激发-收缩偶联起作用。 了解更多
  15. YM-58483

    Catalog No. A16346
    Quick View
    CRAC channel 抑制剂
    YM-58483是CRAC通道和随后的Ca2+信号的第一个选择性抑制剂。 了解更多
  16. Chlorocresol

    Catalog No. A16444
    Quick View
    Chlorocresol是ryanodine受体的活化剂。 了解更多
  17. Cinepazide maleate

    Catalog No. A16454
    Quick View
    Cinepazide maleate是Cinepazide的马来酸盐形式,其为血管扩张剂。 了解更多
  18. Cinnarizine

    Catalog No. A16455
    Quick View
    calcium channel blocker
    Cinnarizine是哌嗪的药物衍生物,其特征在于抗组胺药和钙通道阻滞剂。 了解更多
  19. Aranidipine

    Catalog No. A18291
    Quick View
    Calcium channel antagonist
    Aranidipine (MPC1304) is a Ca2+ channel antagonist with potent and long-lasting antihypertensive effects. 了解更多
  20. ABT-639

    Catalog No. A12330
    Quick View
    T-type Ca2+ channel blocker
    ABT-639 is a novel, peripherally acting, selective T-type Ca2+ channel blocker. 了解更多
  21. Ca2+ channel agonist 1

    Catalog No. A12186
    Quick View
    Ca2+ channel agonist/CDK2 inhibitor
    Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2, with EC50s of 14.23 μM and 3.34 μM, respectively, and is used as a potential treatment for motor nerve terminal dysfunction. 了解更多
  22. Barnidipine

    Catalog No. A21940
    Quick View
    L-type calcium antagonist
    Barnidipine (Mepirodipine) is an L-type calcium antagonist (CaA) with high affinity for [3H] initrendipine binding sites (Ki=0.21 nmol/l), has selective action against CaA receptors. 了解更多
  23. Dantrolene sodium

    Catalog No. A17644
    Quick View
    Calcium channel proteins inhibitor
    Dantrolene sodium is a inhibitor of calcium channel proteins, inhibiting the release of Ca2+ from the sarcoplasm. Dantrolene sodium is a skeletal muscle relaxant which acts by blocking muscle contraction beyond the neuromuscular junction. 了解更多
  24. Tetrandrine (Fanchinine)

    Catalog No. A10921
    Quick View
    Calcium Channel 抑制剂
    Tetrandrine (Fanchinine)是一种钙通道阻滞剂。粉防己碱具有抗炎和抗纤维化作用,使粉防己碱及其相关化合物潜在地用于治疗肺矽肺,肝硬化和类风湿性关节炎。 了解更多
  25. Astragaloside A

    Catalog No. A11405
    Quick View
    Ca2+ signaling modulator
    Astragaloside A是缺氧条件下人脐静脉内皮细胞HIF-1α和通过PI3K/Akt途径血管生成的一种新型调节因子。 了解更多
  26. CK-1827452 (Omecamtiv mecarbil)

    Catalog No. A11206
    Quick View
    Myosin activator
    CK-1827452 (Omecamtiv mecarbil)是选择性的心脏特异性肌球蛋白激活剂。 了解更多
  27. Manidipine 2HCl

    Catalog No. A10554
    Quick View
    Manidipine dihydrochloride是Manidipine的HCl盐形式,Manidipine是Ca2+电流的钙通道阻滞剂,IC50为2.6 nM。 了解更多
  28. Amlodipine

    Catalog No. A10068
    Quick View
    L-type calcium channel blocker
    Amlodipine是一种L型钙通道阻滞剂,具有降压作用。它抑制去极化大鼠主动脉中Ca2 +诱导的收缩(IC50 = 1.9 nM),并在心血管疾病中显示出血管保护作用。 了解更多
  29. Amlodipine besylate (Norvasc)

    Catalog No. A10069
    Quick View
    L-type calcium channel blocker
    Amlodipine besylate是一种L型钙通道阻滞剂,具有降压作用。它抑制去极化大鼠主动脉中Ca2 +诱导的收缩(IC50 = 1.9 nM)。 了解更多
  30. Cilnidipine

    Catalog No. A10215
    Quick View
    Calcium channel blocker
    Cilnidipine是提供血管平滑肌中L型电压门控钙通道和交感神经末梢N型钙通道的双重阻滞剂。 了解更多
  31. Isradipine

    Catalog No. A10487
    Quick View
    calcium channel blocker
    伊拉地平是二氢吡啶类钙通道阻滞剂。 了解更多
  32. Azelnidipine

    Catalog No. A11219
    Quick View
    calcium channel blocker
    Azelnidipine是一种钙阻断剂,可减轻肝纤维化并可能增加抗氧化防御能力。可以减轻肝纤维化并可能增加抗氧化防御能力。 了解更多
  33. Lacidipine

    Catalog No. A11729
    Quick View
    Lacidipine是一种钙通道阻滞剂。 了解更多
  34. Benidipine hydrochloride

    Catalog No. A11730
    Quick View
    Benidipine hydrochloride是一种长效的T型钙通道阻滞剂,对高血压糖尿病患者的血压和肾功能有影响。 了解更多
  35. Nilvadipine (ARC029)

    Catalog No. A11731
    Quick View
    calcium channel blocker
    Nilvadipine (ARC029)是一种钙通道阻滞剂(CCB),用于治疗高血压和慢性主要脑动脉阻塞。 了解更多
  36. Clevidipine

    Catalog No. A11746
    Quick View
    Calcium channel blocker
    Clevidipine是一种二氢吡啶类钙通道阻滞剂,用于在口服治疗不可行或不理想时降低血压。 了解更多
  37. Diethylstilbestrol

    Catalog No. A10309
    Quick View
    Diethylstilbestrol是一种合成的非甾体雌激素,于1938年首次合成。它也被分类为内分泌干扰物。 了解更多
  38. Diltiazem HCl

    Catalog No. A10311
    Quick View
    Diltiazem HCl是一种非二氢吡啶(非DHP)药物,称为钙通道阻滞剂,用于治疗高血压,心绞痛和某些类型的心律不齐。 了解更多
  39. Manidipine (Manyper)

    Catalog No. A10553
    Quick View
    Manidipine (Manyper)是二氢吡啶化合物和钙通道蛋白抑制剂和拮抗剂。 了解更多
  40. Pinaverium Bromide

    Catalog No. A12684
    Quick View
    Pinaverium Bromide是一种痉挛剂,抗胆碱能作用的发生率低。吡那溴铵也是解痉药。 了解更多
  41. Nifedipine

    Catalog No. A10643
    Quick View
    L-type calcium channel blocker.
    Nifedipine是一种L型钙通道阻滞剂。 了解更多
  42. Nimodipine

    Catalog No. A10645
    Quick View
    Calcium Channel 抑制剂
    Nimodipine是一种L型Ca2+通道阻滞剂。 了解更多
  43. BAPTA tetrapotassium

    Catalog No. A13989
    Quick View
    Selective calcium chelator
    BAPTA tetrapotassium是一种选择性钙螯合剂,对Ca2+的亲和力大于Mg2+。 了解更多
  44. BAPTA/AM

    Catalog No. A14023
    Quick View
    Selective calcium chelator
    BAPTA/AM是一种细胞内钙螯合剂,可通过脂氧合酶介导的自由基在小鼠皮层培养物中诱导延迟性坏死。 了解更多
  45. Dantrolene

    Catalog No. A13928
    Quick View
    Ca2+ release 抑制剂
    Dantrolene是一种肌肉松弛剂,其作用可能是通过消除对ryanodine受体的作用来消除肌肉细胞中的兴奋-收缩偶联。 了解更多
  46. Atagabalin

    Catalog No. A13402
    Quick View
    Atagabalin与加巴喷丁相关,加巴喷丁同样与α结合。2β钙通道(1和2)。 了解更多
  47. Berbamine

    Catalog No. A14794
    Quick View
    Calcium channel blocker
    Berbamine是钙通道阻滞剂。 了解更多

47 个项目

每页

设置升序顺序
Rewards