Cell Metabolism
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GW1929
Catalog No. A15099 -
Balaglitazone
Catalog No. A15013 -
BMS-687453
Catalog No. A15836 PPAR 激动剂BMS-687453是一种有效的选择性过氧化物酶体增殖物激活受体(PPAR)α激动剂,对人PPARα的EC(50)为10 nM,在PPAR-GAL4反式激活试验中,选择性是对人PPARgamma的410倍。 了解更多 -
Aleglitazar
Catalog No. A12492 -
Elafibranor
Catalog No. A15454 PPAR 激动剂Elafibranor是过氧化物酶体增殖物激活的受体-α和-δ的激动剂,可诱导非酒精性脂肪性肝炎消退,而不会使纤维化恶化。 了解更多 -
CDDO-Im
Catalog No. A16308 -
5-Aminosalicylic Acid
Catalog No. A10570 PPARγ agonist5-Aminosalicylic acid (Mesalamine) acts as a specific PPARγ agonist and also inhibits p21-activated kinase 1 (PAK1) and NF-κB. 了解更多 -
Pioglitazone hydrochloride
Catalog No. A16670 PPARγ agonistPioglitazone hydrochloride is a potent and selective PPARγ agonist with EC50s of 0.93 and 0.99 μM for human and mouse PPARγ, respectively. 了解更多 -
Fonadelpar
Catalog No. A20848 PPARδ agonistFonadelpar is a PPARδ agonist, used in the research of neuroparalytic keratopathy. 了解更多 -
Tesaglitazar
Catalog No. A20891 PPAR alpha/gamma agonistTesaglitazar is a dual peroxisome proliferator-activated receptor (PPAR) alpha/gamma agonist that is more potent on PPARγ than on PPARα, with EC50s of 13.4 μM and 3.6 μM for rat PPARα and human PPARα, respectively. 了解更多 -
Arhalofenate
Catalog No. A21135 PPARγ agonistArhalofenate (MBX 102) is a selective partial agonist of peroxisome proliferator-activated receptor (PPAR)-γ, used for the treatment of type 2 diabetes. 了解更多 -
Indeglitazar
Catalog No. A21148 PPAR agonistIndeglitazar is an orally available peroxisome proliferator-activated receptor (PPAR) pan-agonist for all three PPAR subtypes alpha (α), delta (δ) and gamma (γ). 了解更多 -
Inolitazone
Catalog No. A21180 PPARγ agonistInolitazone a novel high-affinity PPARγ agonist that is dependent upon PPARγ for its biological activity with IC50 of 0.8 nM for growth inhibition. 了解更多 -
Rosiglitazone maleate
Catalog No. A10809 -
Pioglitazone (Actos)
Catalog No. A11680 PPARγ 激动剂Pioglitazone (Actos)是选择性刺激核受体过氧化物酶体增殖物激活的受体γ(PPAR-γ),并在较小程度上刺激PPAR-α。 了解更多 -
Rosiglitazone (BRL-49653)
Catalog No. A10807 PPAR 激动剂Rosiglitazone (BRL-49653)是有效的降糖药,也是有效的噻唑烷二酮类胰岛素增敏剂,在大鼠,3T3-L1和人体脂肪细胞中IC50分别为12,4和9 nM。Rosiglitazone是PPAR-gamma的配体,对PPAR-alpha没有结合力。 了解更多 -
Troglitazone
Catalog No. A11981 PPARγ 激动剂Troglitazone是一种选择性PPARγ受体激动剂(鼠和人PPARγ受体的EC50值分别为780和555 nM)。 了解更多 -
pirinixic acid (WY 14643)
Catalog No. A12360 -
Inolitazone dihydrochloride
Catalog No. A15129 PPARγ 激动剂Inolitazone dihydrochloride是一种新型的高亲和力PPARγ激动剂,可激活PPARγ,其EC50约为罗格列酮的EC50,对RIE细胞无影响。 了解更多 -
Etofylline
Catalog No. A17491 PPAR agonistEtofylline, also known as BRN-0251760, is a peroxisome proliferator-activated receptor (PPAR) agonist used to treat respiratory and cardiovascular disorders. Etofylline is often used as a bronchodilator. 了解更多 -
Leriglitazone
Catalog No. A18636 PPAR gamma agonistLeriglitazone is a peroxisome proliferator activated receptor (PPAR) gamma agonist. 了解更多 -
Chiglitazar
Catalog No. A12701 PPARα/γ dual agonistChiglitazar is a PPARα/γ dual agonist, with EC50s of 1.2, 0.08, 1.7 μM for PPARα, PPARγ and PPARδ, respectively. 了解更多 -
RGX-104 free Acid
Catalog No. A21513 LXR agonistRGX-104 free Acid is an orally bioavailable and potent liver-X nuclear hormone receptor (LXR) agonist that modulates innate immunity via transcriptional activation of the ApoE gene. 了解更多 -
GW3965 HCl
Catalog No. A11204 -
Sobetirome
Catalog No. A15241 -
SR9238
Catalog No. A15763 -
Cilofexor
Catalog No. A13143 -
Nidufexor
Catalog No. A12625 -
Fexaramine
Catalog No. A21771 FXR agonistFexaramine is a small molecule farnesoid X receptor (FXR) agonist with 100-fold increased affinity relative to natural compounds. 了解更多 -
WAY-362450
Catalog No. A11186 FXR 激动剂WAY-362450是一种高效,选择性和口服可生物利用的法呢类X受体(FXR)激动剂(EC50:4 nM,eff = 149%)。 了解更多 -
Lithocholic acid
Catalog No. A12547 -
Obeticholic Acid
Catalog No. A13866 FXR 激动剂Obeticholic Acid是一种有效的选择性法呢类X受体(FXR)激动剂,EC50为99 nM。 了解更多 -
Px-104
Catalog No. A16999