PDK1

Catalog No.Inhibitor Name PDK-1 Other Targets
A10681OSU-03012
**
A11148BX-795
****
TBK1/IKKɛ,c-Kit,CDK2/CyclinE
A11149BX-912
***
PKA,KDR,CDK2/CyclinE
A11032PHT-427
*
Akt
A12767GSK2334470
***
A12881 BX-517
****
A11511NVP-BAG956
*
PI3K
A13484PS 48
*

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. BX-795

    Catalog No. A11148
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    PDK-1 抑制剂
    BX-795是有效的PDK1抑制剂,可阻断肿瘤细胞中的PDK1/Akt信号传导并抑制培养物中多种肿瘤细胞系的锚定依赖性生长或诱导凋亡。 了解更多
  2. PDK1 inhibitor

    Catalog No. A11528
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    PDK1 抑制剂
    PDK1 inhibitor是PDK1的有效和选择性抑制剂,具有作为抗癌剂的潜力。 了解更多
  3. PDK1 inhibitor

    Catalog No. A16185
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    PDK1 抑制剂
    PDK1 inhibitor,强效,ATP竞争性和选择性双重PI3K和PDPK1抑制剂(PDK1和p-T308-PKB抑制的IC50值分别为34 nM和94 nM。 了解更多
  4. PHT-427

    Catalog No. A11032
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    AKT 抑制剂
    PHT-427是一种新型的Akt/磷脂酰肌醇依赖性蛋白激酶1 pleckstrin同源域抑制剂。 了解更多
  5. OSU-03012

    Catalog No. A10681
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    PDK-1 抑制剂
    OSU-03012 (AR-12)是一种有效的重组PDK-1(phosphoinositide-dependent kinase 1)抑制剂。 了解更多
  6. BX-912

    Catalog No. A11149
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    PDK1 抑制剂
    BX-912是3-磷酸肌醇依赖性激酶1(PDK1)的抑制剂。 了解更多
  7. NVP-BAG956

    Catalog No. A11511
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    PI3K/PDK-1 抑制剂
    NVP-BAG956是一种强效、可逆和ATP竞争性PI3-K/PDK1双激酶抑制剂,对VEGFR 1(IC50 = 2.56 μM)的效力大大降低,对其他15种激酶(IC50 > 10 uM)的活性很小或没有活性。 了解更多
  8. GSK 2334470

    Catalog No. A12767
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    PDK1 抑制剂
    GSK 2334470是一种有效的3-磷酸肌醇依赖性蛋白激酶(PDK1)抑制剂(IC50?10 nM)。 了解更多
  9. PS 48

    Catalog No. A13484
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    PDK1 抑制剂
    PS 48是一种变构磷酸肌醇依赖性蛋白激酶-1(PDK1)激活剂(Kd = 10.3μM)。 了解更多
  10. BX-517

    Catalog No. A12881
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    PDK1 抑制剂
    BX-517是一种有效且选择性的PDK1抑制剂,可与蛋白质的ATP结合袋结合(IC50 = 6 nM)。 了解更多
  11. TEPP-46

    Catalog No. A16279
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    PKM2 activator
    TEPP-46是重组丙酮酸激酶M2(PKM2)的有效选择性活化剂,最大活化浓度(AC50值)的一半为92 nM,相对于PKM1,PKL和PKR几乎没有或没有活性。 了解更多
  12. KPLH1130

    Catalog No. A18494
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    PDK inhibitor
    KPLH1130 is a specific pyruvate dehydrogenase kinase (PDK) inhibitor, blocks macrophage polarization and attenuates proinflammatory responses. KPLH1130 improves glucose tolerance in HFD-fed mice. 了解更多

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