AG-014699 (Rucaparib)

目录号: A10045

PARP inhibitor

AG-014699 (Rucaparib)

AG-014699 (Rucaparib) Chemical Structure

CAS NO. 459868-92-9

AG-014699 (Rucaparib) is a PARP inhibitor that inhibits poly(ADP-ribose) polymerase (PARP) is a key enzyme in DNA repair.

库存: 现货

规格 价格 数量
5 mg
¥ 600.00
25 mg
¥ 2,200.00
50 mg
¥ 3,500.00
100 mg
¥ 5,800.00
10mM * 1mL in DMSO
¥ 1,100.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

生物活性

AG-014699 (Rucaparib) is a PARP inhibitor that inhibits poly(ADP-ribose) polymerase (PARP) is a key enzyme in DNA repair.
Targets
PARP (Cell-free assay)
1.4 nM(Ki)
In vitro (25°C) DMSO 84 mg/mL (199.35 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.73 mL 118.65 mL 237.3 mL
0.5 mM 4.75 mL 23.73 mL 47.46 mL
1 mM 2.37 mL 11.87 mL 23.73 mL
5 mM 0.47 mL 2.37 mL 4.75 mL

*The above data is based on the productmolecular weight 421.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

产品技术资料

目录号 A10045
MECHANISM OF ACTION Inhibitor
M. Wt 421.4
Formula C19H18FN3O.H3PO4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 459868-92-9
Synonyms AG014699, PF-01367338,AG-014447 (as free base)
SMILES CNCC1=CC=C(C=C1)C2=C3CCNC(=O)C4=CC(=CC(=C34)N2)F.OP(=O)(O)O

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