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OSS-128167
Catalog No. A17048 -
Thiomyristoyl
Catalog No. A17166 -
PROTAC Sirt2 Degrader-1
Catalog No. A20005 Sirt2 degraderPROTAC Sirt2 Degrader-1 is a SirReal-based PROTAC, acts as a Sirt2 degrader, composed of a highly potent and isotype-selective Sirt2 inhibitor, a linker, and a bona fide cereblon ligand for E3 ubiquitin ligase. 了解更多 -
SRT 1720 Hydrochloride
Catalog No. A21143 SIRT1 activator ofSRT 1720 Hydrochloride is a selective activator of SIRT1 with an EC50 of 0.10 μM, and shows less potent activities on SIRT2 and SIRT3. 了解更多 -
Sirt2-IN-1
Catalog No. A19348 Sirt2 inhibitorSirt2-IN-1 (Compound 9) is a sirtuin 2 (Sirt2) inhibitor with an IC50 of 163 nM. 了解更多 -
JFD00244
Catalog No. A19517 -
SIRT5 inhibitor 1
Catalog No. A19841 SIRT5 inhibitorSIRT5 inhibitor 1 is a potent Human Sirtuin 5 deacylase inhibitor, with an IC50 of 0.11 μM. 了解更多 -
SirReal1-O-propargyl
Catalog No. A20091 Sirt2 inhibitorSirReal1-O-propargyl is a selective and highly potent Sirtuin 2 (Sirt2) inhibitor, with an IC50 of 2.4 μM. 了解更多 -
GSK 1210151A (I-BET151)
Catalog No. A11783 BET Bromodomain 抑制剂GSK 1210151A (I-BET151)是溴结构域和额外末端（BET）家族蛋白BRD2，BRD3和BRD4的新型选择性抑制剂。 了解更多 -
GSK 525762A (I-BET-762)
Catalog No. A11440 -
Bromosporine
Catalog No. A13163 bromodomain 抑制剂Bromosporine是一种针对溴结构域的广谱抑制剂，对于BRD2，BRD4，BRD9和CECR2的IC50分别为0.41μM，0.29μM，0.122μM和0.017μM。 了解更多 -
UNC 669
Catalog No. A13717 -
(+)-JQ1
Catalog No. A12729 -
OTX015
Catalog No. A13890 -
I-BRD9
Catalog No. A15872 -
(E)-ZL0420
Catalog No. A20136 BRD4 inhibitorZL0420 is a potent and selective bromodomain-containing protein 4 (BRD4) inhibitor with IC50 values of 27 nM against BRD4 BD1 and 32 nM against BRD4 BD2. 了解更多 -
BMS-986158
Catalog No. A19442 Bromodomain inhibitorBMS-986158 is an inhibitor of the bromodomain and extra-terminal (BET) proteins. 了解更多 -
Bromodomain IN-1
Catalog No. A18845 Bromodomain inhibitorBromodomain IN-1 is a Bromodomain inhibitor extracted from patent WO2016069578A1, compound 4 . 了解更多 -
BRD4 Inhibitor-10
Catalog No. A18679 BRD4-BD1 inhibitorBRD4 Inhibitor-10 is a potent BRD4-BD1 inhibitor extracted from patent WO2015022332A1, Compound II-25, has an IC50 of 8 nM. 了解更多
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