Histone Methyltransferase

产品 1 到 50 共 64个

每页
页面:
  1. 1
  2. 2

设置升序顺序
  1. CPI-169

    Catalog No. A15920
    Quick View
    EZH2 抑制剂
    CPI-169是一种有效的选择性EZH2抑制剂,对EZH2 WT,EZH2 Y641N和EZH1的IC50分别为0.24 nM,0.51 nM和6.1 nM。 了解更多
  2. CPI-360

    Catalog No. A15908
    Quick View
    EZH2 抑制剂
    CPI-360是一种有效的,选择性的且具有SAM竞争性的EZH2抑制剂,IC50为102.3 nM,选择性是其他甲基转移酶的100倍以上。 了解更多
  3. Flopropione

    Catalog No. A16550
    Quick View
    5-HT1A receptor antagonist/COMT inhibitor
    Flopropione是5-HT1A受体拮抗剂,也是儿茶酚-邻甲基转移酶(COMT)抑制剂。 了解更多
  4. GSK503

    Catalog No. A15549
    Quick View
    EZH2 抑制剂
    GSK-503是一种有效的EZH2抑制剂,具有潜在的抗癌活性。 了解更多
  5. EPZ011989

    Catalog No. A15544
    Quick View
    EZH2 抑制剂
    EPZ011989是一种有效的,选择性的生物利用型EZH2抑制剂,对于EZH2 wt和EZH2 Y646,Ki <3 nM;选择性是EZH1的15倍,选择性是其他HMTase的3000倍。 了解更多
  6. CM-272

    Catalog No. A17173
    Quick View
    G9a/DNMT 抑制剂
    CM-272是血液恶性肿瘤中针对G9a和DNMT的可逆双重小分子抑制剂。 了解更多
  7. CM-579

    Catalog No. A18692
    Quick View
    G9a/DNMT inhibitor
    CM-579 is a first-in-class reversible, dual inhibitor of G9a and DNMT, with IC50 values of 16 nM, 32 nM for G9a and DNMT, respectively. Has potent in vitro cellular activity in a wide range of cancer cells. 了解更多
  8. SMYD3-IN-1

    Catalog No. A18572
    Quick View
    SMYD3 inhibitor
    SMYD3-IN-1 (compound 29) is an irreversible and selective inhibitor of SMYD3 (SET and MYND domain containing 3), with an IC50 of 11.7 nM. 了解更多
  9. Entacapone

    Catalog No. A10355
    Quick View
    COMT inhibitor
    Entacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment. 了解更多
  10. OICR-9429

    Catalog No. A16641
    Quick View
    Wdr5-MLL interaction antagonist
    OICR-9429 is a novel small-molecule antagonist of the Wdr5-MLL interaction with IC50 of 5 uM. inhibit proliferation and induce differentiation . 了解更多
  11. CPUY074020

    Catalog No. A12190
    Quick View
    G9a inhibitor
    CPUY074020 is a potent G9a inhibitor with an IC50 of 2.18 μM, and possesses anti-proliferative activity . 了解更多
  12. OICR-0547

    Catalog No. A20877
    Quick View
    Wdr5-MLL interaction antagonist
    OICR-0547 is a closely related derivative of OICR-9429. OICR-9429 is a novel small-molecule antagonist of the Wdr5-MLL interaction, while OICR-0547 cannot bind to WDR5. 了解更多
  13. GSK126

    Catalog No. A11757
    Quick View
    EZH2 抑制剂
    GSK126是一种有效的,高选择性的,具有S-腺苷甲硫氨酸竞争性的小分子EZH2甲基转移酶活性抑制剂,可降低总体H3K27me3水平并重新激活沉默的PRC2目标基因。 了解更多
  14. Tolcapone

    Catalog No. A20966
    Quick View
    COMT inhibitor
    Tolcapone (Ro 40-7592) is a selective, potent and orally active COMT inhibitor. 了解更多
  15. MM-102 TFA

    Catalog No. A21941
    Quick View
    WDR5/MLL interaction inhibitor
    MM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide. 了解更多
  16. MM-589 TFA

    Catalog No. A21892
    Quick View
    WDR5 and MLL protein-protein interaction inhibitor
    MM-589 TFA is a potent inhibitor of WD repeat domain 5 (WDR5) and mixed lineage leukemia (MLL) protein-protein interaction. 了解更多
  17. DZNep

    Catalog No. A11377
    Quick View
    EZH2 抑制剂
    3 Deazaneplanocin A(DZNep)是3-deazaadenosine的环戊烯基类似物,最初是作为S-腺苷L-homocysteine水解酶的抑制剂合成的。 了解更多
  18. Entacapone sodium salt

    Catalog No. A21888
    Quick View
    COMT inhibitor
    Entacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment. 了解更多
  19. PF-06821497

    Catalog No. A21388
    Quick View
    EZH2 inhibitor
    PF-06821497 (compound 23a) is a potent, selective and orally active Enhancer of Zeste Homolog 2 (EZH2) inhibitor, with a Ki value <0.1 nM against mutant Y641N EZH2. Exhibits robust tumor growth inhibition. 了解更多
  20. Tazemetostat hydrobromide

    Catalog No. A21759
    Quick View
    EZH2 inhibitor
    Tazemetostat hydrobromide (EPZ-6438 hydrobromide) is a potent, selective and orally available EZH2 inhibitor. 了解更多
  21. UNC-1999

    Catalog No. A13166
    Quick View
    EZH2/EZH1 抑制剂
    UNC-1999是生物可利用抑制剂,对野生型和突变型ezh2以及ezh1具有高体外效力,无细胞试验中IC50分别为2 nM和45 nM,对广泛表观遗传学相关或不相关的靶点选择性大于1000倍。 了解更多
  22. GSK2807 Trifluoroacetate

    Catalog No. A21731
    Quick View
    SMYD3 inhibitor
    GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM. 了解更多
  23. EI1

    Catalog No. A12711
    Quick View
    EZH2 抑制剂
    EI1是EZH2的一种有效的选择性小分子抑制剂,野生型EZH2和EZH2 Y641F突变体的IC50值分别为15 nM和13 nM。 了解更多
  24. AZ505

    Catalog No. A13061
    Quick View
    SMYD2 抑制剂
    AZ505是一种有效且高度选择性的致癌蛋白SMYD2抑制剂(IC50 = 0.12μM),具有潜在的抗癌活性,是SMYD3(IC50> 83.3μM)的600倍以上; DOT1L(IC50> 83.3μM); EZH2(IC50> 83.3μM)。 了解更多
  25. AZ505 ditrifluoroacetate

    Catalog No. A13169
    Quick View
    SMYD2 抑制剂
    AZ505 ditrifluoroacetate是一种有效且高度选择性的致癌蛋白SMYD2抑制剂(IC50 = 0.12 uM),具有潜在的抗癌活性,是SMYD3的> 600倍(IC50> 83.3 uM)。DOT1L(IC50> 83.3 uM);EZH2(IC50> 83.3 uM)。 了解更多
  26. CPI-1205

    Catalog No. A16357
    Quick View
    EZH2 抑制剂
    CPI-1205是高效的(生化IC50 = 0.002μM,细胞EC50 = 0.032μM)和EZH2的选择性抑制剂。 了解更多
  27. MI-503

    Catalog No. A20975
    Quick View
    menin-mLL interaction inhibitor
    MI-503 is a highly potent and orally bioavailable small molecule inhibitor of the menin-mLL interaction. 了解更多
  28. EPZ031686

    Catalog No. A16375
    Quick View
    SMYD3/ MEKK2 抑制剂
    EPZ031686是SMYD3和MEKK2的非竞争性抑制剂,Ki = 1.2和1.1 nM。 了解更多
  29. JQEZ5

    Catalog No. A16961
    Quick View
    EZH2 抑制剂
    JQEZ5是一种有效的选择性SAM竞争性EZH2赖氨酸甲基转移酶抑制剂,IC50值为11 nM。 了解更多
  30. PF-06726304

    Catalog No. A16937
    Quick View
    EZH2 抑制剂
    PF-06726304是一种有效且与SAM竞争的EZH2(Zeste Homolog 2的增强剂)赖氨酸甲基转移酶抑制剂。 了解更多
  31. JNJ-64619178

    Catalog No. A16861
    Quick View
    Histone Methyltransferase 抑制剂
    JNJ-64619178是PRMT5抑制剂,在不同的体外和细胞条件下均具有高选择性和强效性(亚纳摩尔范围,PRMT5-MEP-50 IC50 = 0.14 nM),并具有良好的药代动力学和安全性。 了解更多
  32. BAY-598

    Catalog No. A17012
    Quick View
    SMYD2 抑制剂
    BAY-598是用于SMYD2的强效,具有肽竞争性的化学探针。 了解更多
  33. GNA002

    Catalog No. A13266
    Quick View
    EZH2 inhibitor
    GNA002 is a highly potent, specific and covalent EZH2 (Enhancer of zeste homolog 2) inhibitor with an IC50 of 1.1 μM. 了解更多
    • 最新产品

    BCI-121

    Catalog No. A17065
    Quick View
    SMYD3 抑制剂
    BCI-121是SMYD3抑制剂。它通过削弱癌细胞的生长来发挥作用。 了解更多
  34. BIX-01338 hydrate

    Catalog No. A21812
    Quick View
    histone lysine methyltransferase inhibitor
    BIX-01338 hydrate is a histone lysine methyltransferase inhibitor. 了解更多
  35. BIX 01294

    Catalog No. A11763
    Quick View
    G9a/GLP HMT 抑制剂
    BIX 01294是一种G9a样蛋白和G9a组蛋白赖氨酸甲基转移酶抑制剂。 了解更多
  36. EPZ-5676 (Pinometostat)

    Catalog No. A12735
    Quick View
    DOT1L 抑制剂?
    EPZ-5676 (Pinometostat)是组蛋白甲基转移酶的小分子抑制剂,具有潜在的抗肿瘤活性。 了解更多
  37. Chaetocin

    Catalog No. A12812
    SUV39H HMT 抑制剂
    Chaetocin是组蛋白甲基转移酶SUV39H1抑制剂(IC50 = 0.8μM)。在体外诱导骨髓瘤细胞系的凋亡; 在小鼠骨髓瘤模型中具有抗增殖活性。 了解更多
  38. UNC0646

    Catalog No. A13194
    Quick View
    G9a/GLP HMTase 抑制剂
    UNC0646是一种有效且选择性的同源蛋白赖氨酸甲基转移酶G9a和GLP抑制剂(G9a和GLP的IC50值分别为6 nM和15 nM)。 了解更多
  39. UNC0631

    Catalog No. A13195
    Quick View
    G9a 抑制剂
    UNC-0631是一种新型G9a抑制剂,在多种细胞系中均具有出色的效能,并且功能性效能与细胞毒性的分离效果极佳。 了解更多
  40. GSK343

    Catalog No. A13114
    Quick View
    EZH2 抑制剂
    GSK343是有效的组蛋白H3-赖氨酸27(H3K27)甲基转移酶EZH2抑制剂(IC = 4 nM)。对除EZH1以外的其他HMT的选择性是1000倍(选择性是60倍)。GSK343抑制HCC1806细胞中的H3K27甲基化,IC小于200nM(通过免疫荧光测量)。 了解更多
  41. Opicapone (BIA 9-1067)

    Catalog No. A13110
    Quick View
    COMT 抑制剂
    Opicapone (BIA 9-1067)是一种新型邻苯二酚-o-甲基转移酶抑制剂。 了解更多
  42. UNC0321

    Catalog No. A13200
    Quick View
    G9a HMTase 抑制剂
    UNC0321是第一种具有皮摩尔效价的G9a抑制剂,也是迄今为止最有效的G9a抑制剂。 了解更多
  43. EPZ-6438 (Tazemetostat)

    Catalog No. A12712
    Quick View
    EZH2 抑制剂
    EPZ-6438 (Tazemetostat)是一种有效的,选择性的,口服可利用的EZH2酶促活性小分子抑制剂,无细胞试验中Ki 和 IC50分别为2.5 nM 和 11 nM。它诱导SMARCB1缺失的MRT细胞中的凋亡和分化。 了解更多
  44. EPZ004777

    Catalog No. A12983
    Quick View
    DOT1L 抑制剂
    EPZ004777是dot1l的有效选择性抑制剂。epz004777选择性抑制细胞h3k79甲基化并抑制关键mll融合靶基因的表达。 了解更多
  45. SGC 0946

    Catalog No. A12941
    Quick View
    DOT1L 抑制剂
    SGC 0946是有效的DOT1L甲基转移酶抑制剂,可阻断A431细胞和MCF10A细胞中的H3K79甲基化。 了解更多
  46. UNC 0638

    Catalog No. A13690
    Quick View
    G9a/GLP 抑制剂
    UNC 0638是G9a和GLP组蛋白赖氨酸甲基转移酶的选择性抑制剂。 了解更多
  47. MI-3

    Catalog No. A14218
    Quick View
    menin-MLL interaction 抑制剂
    MI-3是一种有效的Menin-MLL相互作用抑制剂,IC50为648 nM。 了解更多
  48. PFI-2

    Catalog No. A14216
    Quick View
    SETD7 抑制剂
    PFI-2是一种有效的,选择性的,具有细胞活性的赖氨酸甲基转移酶SETD7抑制剂,Ki(app)和IC50为0.33 nM和2 nM,选择性是其他甲基转移酶和其他非表观遗传靶标的1000倍。 了解更多
  49. MM-102

    Catalog No. A14315
    Quick View
    MLL1 抑制剂
    MM-102是一种高亲和力的拟肽MLL1抑制剂,IC50为0.4 uM。 了解更多

产品 1 到 50 共 64个

每页
页面:
  1. 1
  2. 2

设置升序顺序
Rewards