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Cell Cycle

产品 51 到 100 共 257个

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  1. PD 0332991 Isethionate
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    PD 0332991 Isethionate

    Catalog No. A13811
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    CDK4/6 抑制剂
    PD 0332991 Isethionate是CDK4/6的高选择性抑制剂，IC50分别为11 nM/16 nM。 了解更多
  2. P276-00
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    P276-00

    Catalog No. A13547
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    CDK 抑制剂
    P276-00是一种新型CDK1，CDK4和CDK9抑制剂，IC50分别为79 nM，63 nM和20 nM。在第2/3阶段。 了解更多
  3. LEE011 (Ribociclib)
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    LEE011 (Ribociclib)

    Catalog No. A13549
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    CDK4/6 抑制剂
    LEE011 (Ribociclib)是一种可口服的细胞周期蛋白依赖性激酶（CDK）抑制剂，靶向细胞周期蛋白D1/CDK4和细胞周期蛋白D3/CDK6细胞周期途径，具有潜在的抗肿瘤活性。 了解更多
  4. LDC000067
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    LDC000067

    Catalog No. A14273
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    CDK 抑制剂
    LDC000067是一种高选择性CDK9抑制剂。 了解更多
  5. AMG-925
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    AMG-925

    Catalog No. A14025
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    Dual FLT3/CDK4 抑制剂
    AMG-925是一种有效，选择性和生物利用性的FLT3/细胞周期蛋白依赖性激酶4（CDK4）双激酶抑制剂。 了解更多
  6. CVT-313
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    CVT-313

    Catalog No. A15054
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    CDK2 抑制剂
    CVT-313是一种有效，选择性，可逆且具有ATP竞争性的CDK2抑制剂（对于Cdk2/A和Cdk2/E，IC50 = 0.5 uM；对于Cdk1/B为4.2 uM；对于Cdk4/D1为215 uM）。 了解更多
  7. Purvalanol A
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    Purvalanol A

    Catalog No. A15517
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    CDK 抑制剂
    Purvalanol A是一种有效的细胞渗透性细胞周期蛋白依赖性蛋白激酶（cdk）抑制剂。对于cdc2/cyclin B，cdk2/cyclin A，cdk2/cyclin E，cdk4/cyclin D1和cdk5-p35，IC50值分别为4、70、35、850和75 nM。 了解更多
  8. NVP-LCQ195
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    NVP-LCQ195

    Catalog No. A15196
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    CDK 抑制剂
    NVP-LCQ195是CDK1，CDK2，CDK3和CDK5的小分子杂环抑制剂，IC50为1-42 nM。 了解更多
  9. AG-024322
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    AG-024322

    Catalog No. A15485
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    CDK 抑制剂
    AG-24322是第二代CDK抑制剂。AG-024322是有效的CDK1，CDK2和CDK4抑制剂，可在临床前模型中产生细胞周期停滞和抗肿瘤活性。 了解更多
  10. NU2058
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    NU2058

    Catalog No. A15767
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    CDK 抑制剂
    NU2058是基于鸟嘌呤的CDK抑制剂，对CDK2和CDK1的IC50为17 uM和26 uM。 了解更多
  11. CDK8-IN-1
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    CDK8-IN-1

    Catalog No. A12961
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    CDK8 inhibitor
    CDK8-IN-1 is a potent and selective CDK8 inhibitor with an IC50 of 3 nM. 了解更多
  12. CDK-IN-2
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    CDK-IN-2

    Catalog No. A11353
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    CDK9 inhibitor
    CDK-IN-2 is a potent and specific CDK9 inhibitor with IC50 of <8 nM, extracted from reference 1, example 4. 了解更多
  13. Senexin A
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    Senexin A

    Catalog No. A21166
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    CDK8 inhibitor
    Senexin A is a CDK8 inhibitor with an IC50 of 280 nM. 了解更多
  14. Voruciclib hydrochloride
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    Voruciclib hydrochloride

    Catalog No. A21385
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    CDK inhibitor
    Voruciclib hydrochloride is a clinical stage orally active and selective CDK inhibitor with Ki values of 0.626 nM-9.1 nM. 了解更多
  15. PHA-767491 hydrochloride
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    PHA-767491 hydrochloride

    Catalog No. A21395
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    dual Cdc7/Cdk9 inhibitor
    PHA-767491 hydrochloride is a dual Cdc7/Cdk9 inhibitor, with IC50s of 10 nM and 34 nM, respectively. 了解更多
  16. CDKI-73
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    CDKI-73

    Catalog No. A21467
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    CDK9 inhibitor
    CDKI-73 is a potent CDK9 inhibitor with Ki of 4 nM; shows selective toxicity to CLL cells(LD50=80 nM) versus normal B cell and normal CD34+ cell(LD50>20 uM). 了解更多
  17. CDK9-IN-1
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    CDK9-IN-1

    Catalog No. A21552
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    CDK9 inhibitor
    CDK9-IN-1 is a novel, selective CDK9 inhibitor for the treatment of HIV infection, with an IC50 of 39 nM for CDK9/CycT1, extracted from reference, compound 87. 了解更多
  18. (±)-BAY-1251152
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    (±)-BAY-1251152

    Catalog No. A21564
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    PTEF/CDK9 inhibitor
    (±)-BAY-1251152 is a racemic mixture of BAY-1251152. BAY-1251152 is a potent and highly selective PTEF/CDK9 inhibitor. 了解更多
  19. (-)-BAY-1251152
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    (-)-BAY-1251152

    Catalog No. A21570
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    PTEF/CDK9 inhibitor
    (-)-BAY-1251152 is an enanthiomer of BAY-1251152 with rotation (-). BAY-1251152 is a potent and highly selective PTEF/CDK9 inhibitor. 了解更多
  20. Lerociclib dihydrochloride
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    Lerociclib dihydrochloride

    Catalog No. A21577
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    CDK4/CDK6 inhibitor
    Lerociclib dihydrochloride (G1T38 dihydrochloride) is a potent and selective inhibitor of CDK4/CDK6, with IC50s of 1 nM and 2 nM for CDK4/CyclinD1 and CDK6/CyclinD3, respectively. 了解更多
  21. LDC4297
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    LDC4297

    Catalog No. A21613
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    CDK7 inhibitor
    LDC4297 is a potent and selective CDK7 inhibitor with an IC50 of 0.13 nM. 了解更多
  22. BS-181 hydrochloride
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    BS-181 hydrochloride

    Catalog No. A21988
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    CDK7 inhibitor
    BS-181 hydrochloride is a highly selective CDK7 inhibitor with IC50 of 21 nM, and > 40-fold selective for CDK7 than CDK1, 2, 4, 5, 6, or 9. 了解更多
  23. SEL120-34A HCl
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    SEL120-34A HCl

    Catalog No. A21485
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    CDK8 inhibitor
    SEL120-34A HCl is a potent, selective, orally available, ATP-competitive CDK8 inhibitor, with IC50s of 4.4 nM and 10.4 nM for CDK8/CycC and CDK19/CycC, respectively, with antitumor activity. 了解更多
  24. NU6300
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    NU6300

    Catalog No. A21025
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    ATP-competitive CDK2 inhibitor
    NU6300 is the first covalent ATP-competitive CDK2 inhibitor. 了解更多
  25. Indirubin
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    Indirubin

    Catalog No. A10471
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    CDK & GSK-3β 抑制剂
    Indirubin是中国抗白血病药物的活性成分，是一种有效的细胞周期蛋白依赖性激酶和GSK-3β抑制剂，IC50约为5 μM和0.6 μM。 了解更多
  26. SNS-032 (BMS-387032)
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    SNS-032 (BMS-387032)

    Catalog No. A10850
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    CDK 抑制剂
    SNS-032（BMS-387032）是细胞周期蛋白依赖性激酶（Cdks）2、7和9的高度选择性和有效抑制剂，具有体外生长抑制作用，并具有诱导恶性B细胞凋亡的能力。 了解更多
  27. AT7519
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    AT7519

    Catalog No. A10093
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    CDK 抑制剂
    AT7519是多种细胞周期蛋白依赖性激酶（CDK）的抑制剂，可导致细胞周期停滞，诱导细胞凋亡和抑制肿瘤细胞增殖。作用于CDK1，2，4，6和9时，IC50为10-210 nM，对CDK3作用效果稍弱，对CDK7几乎没有抑制活性。 了解更多
  28. BS-181
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    BS-181

    Catalog No. A10163
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    CDK 抑制剂
    BS-181 是作为CDK7抑制剂的潜在抗肿瘤剂。 了解更多
  29. Flavopiridol HCl
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    Flavopiridol HCl

    Catalog No. A11045
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    CDK 抑制剂
    Flavopiridol HCl是细胞周期蛋白依赖性激酶的抑制剂。（-）-顺式形式诱导特定肿瘤细胞的凋亡。 了解更多
  30. JNJ-7706621
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    JNJ-7706621

    Catalog No. A10494
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    CDK/Aurora A/B 抑制剂
    JNJ-7706621是对CDK1/2具有最高效力的pan-CDK抑制剂，IC50为9 nM/4 nM，并且在无细胞分析中对CDK1/2的选择性是CDK3/4/6的6倍以上。它还能有效抑制极光A/B，对Plk1和Wee1没有活性。 了解更多
  31. PHA-848125 (Milciclib)
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    PHA-848125 (Milciclib)

    Catalog No. A11047
    CDK 抑制剂
    PHA-848125 (Milciclib)是一种有效的，ATP竞争性CDK抑制剂，作用于CDK2，IC50为45 nM，作用于CDK2比作用于CDK1，2，4，5和7选择性高3倍以上。 了解更多
  32. AZD5438
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    AZD5438

    Catalog No. A11105
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    CDK 抑制剂
    AZD5438是有效的细胞周期蛋白依赖性激酶（CDK）1、2和9抑制剂（IC50值分别为16、6和20 nM）。 了解更多
  33. BMS-265246
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    BMS-265246

    Catalog No. A11154
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    CDK 抑制剂
    BMS-265246是cdk2/cyclin E和cdk1/cyclin B以及cdk4/cyclin D的强新吡唑并吡啶抑制剂。 了解更多
  34. R547
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    R547

    Catalog No. A11190
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    CDK 抑制剂
    R547是一种新型的细胞周期和转录周期依赖性激酶（CDKs）选择性抑制剂（CDK1，CDK2和CDK4分别为Ki = 1、3和1 nM），具有出色的体外细胞效价，可抑制各种细胞的生长。人肿瘤细胞系。 了解更多
  35. AT7519 HCl
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    AT7519 HCl

    Catalog No. A11313
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    CDK 抑制剂
    AT7519是多种细胞周期蛋白依赖性激酶（CDK）的抑制剂，可导致细胞周期停滞，诱导细胞凋亡和抑制肿瘤细胞增殖。 了解更多
  36. CGP60474
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    CGP60474

    Catalog No. A11347
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    CDK 抑制剂
    CGP60474是细胞周期蛋白依赖性激酶(CDK)的有效抑制剂。 了解更多
  37. Purvalanol B
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    Purvalanol B

    Catalog No. A12352
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    CDK 抑制剂
    Purvalanol B是一种细胞周期蛋白依赖性激酶抑制剂。对于cdc2/cyclin B，cdk2/cyclin A，cdk2/cyclin E，cdk4/cyclin D1和cdk5-p35的ic50值分别为6、6、9、> 10，000和6 nm。对一系列其他蛋白激酶具有选择性(IC50 > 10，000 nM)。 了解更多
  38. NU 6102
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    NU 6102

    Catalog No. A12438
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    CDK 抑制剂
    NU 6102与CDK4/D1（IC50 = 1.6μM），DYRK1A（IC50 = 0.9μM），PDK1（IC50 = 0.8μM）和ROCKII（IC50 = 0.6μM）相比，NU6102对CDK1和CDK2具有选择性。 了解更多
  39. Wogonin
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    Wogonin

    Catalog No. A12216
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    CDK9 抑制剂
    Wogonin是抗炎剂和CDK9抑制剂，并且在抑制CDK9活性的剂量下不抑制CDK2, CDK4和CDK6也抑制N-乙酰转移酶。 了解更多
  40. TG003
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    TG003

    Catalog No. A13721
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    Clk 抑制剂
    TG003是Cdc2样激酶（Clk）的有效，特异性，可逆和ATP竞争性抑制剂。 了解更多
  41. THZ1
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    THZ1

    Catalog No. A14192
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    CDK7 抑制剂
    THZ1是一种新型的选择性强效共价CDK7抑制剂，IC50（结合亲和力）为3.2 nM。抑制Jurkat细胞的增殖，IC50为50 nM。 了解更多
  42. TG-02 (SB1317)
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    TG-02 (SB1317)

    Catalog No. A11962
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    FLT3 抑制剂
    TG-02 (SB1317)是一种新型的小分子有效CDK/JAK2/FLT3抑制剂。 了解更多
  43. NU6027
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    NU6027

    Catalog No. A14136
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    ATR/CDK 抑制剂
    NU6027是一种有效的细胞ATR活性抑制剂（IC（50）=6.7μM），并以ATR依赖的方式增强羟基脲和顺铂的细胞毒性。 了解更多
  44. ML167
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    ML167

    Catalog No. A14297
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    Clk4 抑制剂
    ML167是一种高度选择性的Cdc2样激酶4（Clk4）抑制剂。 了解更多
  45. SU9516
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    SU9516

    Catalog No. A14318
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    CDK2 抑制剂
    SU9516是一种有效的选择性cdk2抑制剂。它抑制pRb磷酸化，导致增强的pRB/E2F复合物形成，并诱导G1和G2-M细胞周期停滞。 了解更多
  46. Voruciclib
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    Voruciclib

    Catalog No. A14392
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    CDK 抑制剂
    Voruciclib是一种黄酮和细胞周期蛋白依赖性激酶（CDK）抑制剂，具有潜在的抗肿瘤活性。 了解更多
  47. CA-224
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    CA-224

    Catalog No. A14414
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    CDK4 抑制剂
    CA-224是有效的CDK4抑制剂，也是fascaplysin的非平面类似物，在体外特异性抑制Cdk4-cyclin D1。 了解更多
  48. Ro 3306
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    Ro 3306

    Catalog No. A14437
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    CDK1 抑制剂
    Ro 3306是一种具有ATP竞争能力的有效细胞周期蛋白依赖性激酶（cdk）1抑制剂（cdk1/cyclin B1和cdk1/cyclin A的Ki值分别为35和110 nM。 了解更多
  49. PHA690509
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    PHA690509

    Catalog No. A13550
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    CDK 抑制剂
    PHA690509是ATP竞争性CDK抑制剂。 了解更多
  50. AZD5597
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    AZD5597

    Catalog No. A13506
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    CDK 抑制剂
    AZD5597是有效的CDK抑制剂，对一系列癌细胞具有体外抗增殖作用。 了解更多

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  1. Chk (38)
  2. CDK (97)
  3. Aurora Kinase (37)
  4. PLK (14)
  5. ROCK (33)
  6. c-Myc (5)
  7. Wee1 (2)
  8. Ras (38)
  9. DYRK (11)
  10. G-quadruplex (3)
  11. RAD51 (3)
作用机制
  1. Inhibitor (抑制剂) (250)
  2. Agonist (激动剂) (1)
  3. Antagonist (拮抗剂) (1)
  4. Activator (激活剂) (2)
  5. Degrader (降解剂) (1)
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  1. A3 adenosine receptor (1)
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  5. Aurora C (11)
  6. Bcr-Abl (1)
  7. CDK (3)
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  10. Chk2 (1)
  11. CYP3A4 (1)
  12. FAK (1)
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  23. PDE3 (1)
  24. PDGFRβ (1)
  25. RET (1)
  26. Src (3)
  27. TrkA (2)
  28. VEGFR2 (FLK1) (2)
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