c-Kit

Catalog No.Inhibitor Name c-KitOther
A10290Dasatinib
***
Abl,Src
A10468Imatinib Mesylate
**
PDGFR,v-Abl
A10996Cabozantinib
***
VEGFR2/KDR,c-Met,VEGFR3/FLT4
A10103Axitinib
****
VEGFR1/FLT1,VEGFR2/Flk1,VEGFR2/KDR
A10699Pazopanib HCl
*
VEGFR1,VEGFR2,VEGFR3
A11411Dovitinib
****
FLT3,FGFR1,VEGFR3/FLT4
A10967Vatalanib 2HCl
*
VEGFR2/KDR,VEGFR1/FLT1,VEGFR2/Flk1
A10558Masitinib
*
Lyn B,PDGFRα,PDGFRβ
A10101Tivozanib
**
VEGFR2,VEGFR3,EphB2
A10610Amuvatinib
***
PDGFRα (V561D),FLT3 (D835Y)
A10608Motesanib Diphosphate
***
VEGFR1,VEGFR2,VEGFR2/Flk1
A10679OSI-930
**
FLT1,KDR,CSF-1R
A10502Ki8751
**
VEGFR2,PDGFRα,FGFR2
A10903Telatinib
****
VEGFR3,VEGFR2,PDGFRα
A11518Pazopanib
*
VEGFR1,VEGFR2,VEGFR3
A10198Dovitinib Dilactic Acid
****
FLT3,FGFR1,VEGFR3/FLT4
A16320Dasatinib Monohydrate
***
Abl ,Src
A14156AZD2932
***
PDGFRβ,Flt3,VEGFR-2
A10880Sunitinib Malate
FLT3,PDGFRβ,VEGFR2
A15062DCC-2618
***
PDGFRα, PDGFRβ
A15519PLX647
***
Fms
A15520Pexidartinib (PLX3397)
***
CSF-1R, Flt-3

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. Ki8751

    Catalog No. A10502
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    VEGFR-2 抑制剂
    ki8751是一种细胞可渗透的喹啉氧基苯基脲化合物,在基于细胞和无细胞的检测中起Flk-1 (VEGFR-2)选择性抑制剂的作用。 了解更多
  2. AC710

    Catalog No. A15933
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    FLT3/KIT/PDGFRα/PDGFRβ 抑制剂
    AC710是一种有效的,具有活性的,选择性血小板衍生的生长因子受体家族激酶抑制剂,具有潜在的抗癌活性。 了解更多
  3. Pazopanib (GW-786034)

    Catalog No. A11518
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    VEGFR 抑制剂
    Pazopanib (GW-786034)是VEGFR-1,VEGFR-2,VEGFR-3,PDGFR-a/β和c-kit的有效且选择性的多靶点酪氨酸激酶抑制剂,可阻止肿瘤生长并抑制血管生成。 了解更多
  4. AC710 Mesylate

    Catalog No. A16246
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    FLT3/KIT/PDGFRα/PDGFRβ 抑制剂
    AC710 Mesylate是一种有效的选择性PDGFR家族激酶抑制剂,对于FLT3/KIT/PDGFRα/PDGFRβ的Kd值分别为0.6 nM/1.0 nM/1.3 nM/1.0 nM。 了解更多
  5. Masitinib mesylate

    Catalog No. A15152
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    KIT/PDGFR 抑制剂
    Masitinib mesylate是Kit和PDGFRα/β的新型抑制剂,IC50为200 nM和540 nM/800 nM,对ABL和c-Fms的抑制作用较弱。 了解更多

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