GSK126

促销

EZH2 抑制剂

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产品目录号: A11757

库存状态:中国现货中国现货

产品名 目录号 价格 数量
GSK126 2mg A11757-2
¥ 400.00
GSK126 5mg A11757-5
¥ 600.00
GSK126 10mg A11757-10
¥ 900.00
GSK126 25mg A11757-25
¥ 1,600.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

GSK126 is a potent, highly selective, S-adenosyl-methionine-competitive, small-molecule inhibitor of EZH2 methyltransferase activity, decreases global H3K27me3 levels and reactivates silenced PRC2 target genes.

GSK126

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Chemical Information

目录号 A11757
Mechanism of action Inhibitor
分子量 526.67
化学分子式 C31H38N6O2
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 1346574-57-9
Synonyms GSK 126, GSK-126
SMILES code CC[C@H](C)N1C=C(C2=C(C=C(C=C21)C3=CN=C(C=C3)N4CCNCC4)C(=O)NCC5=C(C=C(NC5=O)C)C)C
化学名称 (S)-1-(sec-butyl)-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide

Biological Activity

Description
GSK126 is a potent, highly selective, S-adenosyl-methionine-competitive, small-molecule inhibitor of EZH2 methyltransferase activity, decreases global H3K27me3 levels and reactivates silenced PRC2 target genes.
Targets
EZH2
9.9 nM

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