“angiotensin converting enzyme ace”的搜索结果
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angiotensin 1 (AT1) and AT2 receptor agonist
Angiotensin III is an angiotensin 1 (AT1) and AT2 receptor agonist.
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angiotensin-converting enzyme inhibitor
Lisinopril (MK-521) is angiotensin-converting enzyme inhibitor, used in treatment of hypertension, congestive heart failure, and heart attacks.
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ACE inhibitor
Rentiapril is an orally active angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.
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ACE inhibitor
Utibapril is an angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activities.
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ACE inhibitor
NCX899 is a NO-releasing derivative of enalapril, and shows inhibitory activity against angiotensin-converting enzyme (ACE) activity.
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ACE inhibitor
Imidaprilate is an active metabolite of TA-6366, acts as a potent angiotensin converting enzyme (ACE) inhibitor, with an IC50 of 2.6 nM, and is used in the research of hypertensive disease.
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ACE inhibitor
Zofenopril is an angiotensin-converting enzyme (ACE) inhibitor with an IC50 of 81 μM.
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ACE inhibitor
H-Val-Pro-Pro-OH, a milk-derived proline peptides derivative, is an inhibitor of Angiotensin I converting enzyme (ACE), with an IC50 of 9 μM.
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Angiotensin II human is a vasoconstrictor that acts on the AT1 and the AT2 receptor.
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Angiotensin 1/2 + A (2 - 8)有效的内源性血管收缩肽;血管紧张素(Ang)的衍生物II。
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Angiotensin 1/2 (1-6)是一种包含氨基酸1-6的肽,是从血管紧张素I/II肽转化而来的。
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Angiotensin 1/2 (1-5)是一种包含氨基酸1-5的肽,是从血管紧张素I/II转化而来的。
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Angiotensin 1/2 (1-9)是一种肽(ASP-ARG-VAL-TYR-ILE-HIS-PRO-PHE-HIS),包含从血管紧张素I/II肽转换而来的氨基酸1-9。
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Angiotensin III (human,mouse)是在血管紧张素II的N末端裂解形成的六肽,血管紧张素II是位于红细胞和大多数组织血管床中的血管紧张素酶在肾素-血管紧张素-醛固酮(RAAS)系统中的关键因素。
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Angiotensin II是一种八肽激素,在心血管稳态中起着核心作用。
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Angiotensin (1-7)是一种内源性肽片段,可以分别通过内切肽酶或羧肽酶从Ang I或Ang II产生。
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H-Ile-Pro-Pro-OH, a milk-derived peptide, inhibits angiotensin-converting enzyme (ACE)with an IC50 of 5 μM. Antihypertensive tripeptides.
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non-peptide angiotensin II receptor antagonist
Fimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys.
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ME1 inhibitor
Malic enzyme inhibitor ME1 (ME1; compound 1) is a potent inhibitor of Malic enzyme (ME1) with an IC50 of 0.15 μM.
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Angiotensin II receptor antagonist
Losartan is an angiotensin II receptor antagonist, competing with the binding of angiotensin II to AT1 receptors with IC50 of 20 nM.
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Angiotensin I (human,mouse,rat)是由肾素对血管紧张素原的作用形成的。
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ACE/NEP inhibitor
Omapatrilat is a dual inhibitor of the metalloproteases ACE and NEP with Ki values of 0.64 and 0.45 nM, respectively.
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ACE 抑制剂
Ramipril是一种血管紧张素转化酶(ACE)抑制剂,IC50为5 nM。
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ACE 抑制剂
Enalapril maleate是一种血管紧张素转换酶(ACE)抑制剂,用于治疗高血压和某些类型的慢性心力衰竭。
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ACE 抑制剂
Fosinopril sodium是一种血管紧张素转换酶(ACE)抑制剂,用于治疗高血压和某些类型的慢性心力衰竭。
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ECE inhibitor
(±)-WS75624B is an endothelin converting enzyme (ECE) inhibitor with an IC50 of 0.03 μg/mL.
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dual TACE/MMPs inhibitor
Apratastat is an orally active, potent, and reversible dual inhibitor of tumor necrosis factor-α converting enzyme (TACE) and matrix metalloproteinases (MMPs) .
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angiotensin II receptor antagonist
EMD-66684 is a non-peptide angiotensin II receptor antagonist.
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nonpeptide angiotensin II receptor antagonist
L-159282 is a highly potent, orally active, nonpeptide angiotensin II receptor antagonist, with anti-hypertensive activity.
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angiotensin AT1 receptor antagonist
L162389 is a potent antagonist of angiotensin AT1 receptor with Ki of 28 nM.
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angiotensin II receptor antagonist
CGP48369 is a nonpeptidic angiotensin II receptor antagonist, used for anti-hypertensive research.
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angiotensin II receptor antagonist
Pratosartan is a selective angiotensin II receptor antagonist.
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angiotensin-(1-7) receptor agonist
AVE 0991 is a nonpeptide and orally active angiotensin-(1-7) receptor agonist with an IC50 of 21 nM.
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angiotensin II type 1 receptor antagonist
Azilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist.
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angiotensin II receptor antagonist
Losartan D4 Carboxylic Acid is the deuterium labeled Losartan(EXP-3174), which is an angiotensin II receptor antagonist.
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Angiotensin-II subtype 2 receptor(AT2 R) agonist
CGP-42112(CGP-42112A) is a potent Angiotensin-II subtype 2 receptor(AT2 R) agonist.
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angiotensin II and endothelin A receptor antagonist
Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively.
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angiotensin II receptor type 1 antagonist
Azilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.
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angiotensin II receptor antagonist
Valsartan (CGP-48933) is an angiotensin II receptor antagonist for the treatment of high blood pressure and heart failure.
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Angiotensin AT1 receptor antagonist
SL910102 is a nonpeptide angiotensin AT1 receptor antagonist.
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anti-tumor agent
Sinapinic acid (Sinapic acid) is a phenolic compound isolated from Hydnophytum formicarum Jack. Rhizome, acts as an inhibitor of HDAC, with an IC50 of 2.27 mM, and also inhibits ACE-I activity. Sinapinic acid posssess potent anti-tumor activity, induces apoptosis of tumor cells.
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Immunomodulator
Aceneuramic acid hydrate是潜在地用于治疗遗传性包涵体肌病(HIBM)的免疫调节剂。
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Enkephalin-degrading and ACE 抑制剂
Spinorphin是一种内源性因子,对脑啡肽降解酶具有抑制作用。
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ACE 抑制剂
Zofenopril calcium是一种血管紧张素转化酶ACE抑制剂。
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- Tomas Jasenovec, .et al. Angiotensin System Modulations in Spontaneously Hypertensive Rats and Consequences on Erythrocyte Properties; Action of MLN-4760 and Zofenopril, Biomedicines, 2021, Dec 14;9(12):1902 PMID: 34944718
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Imidapril (Tanatril)是血管紧张素转化酶(ACE)的抑制剂。
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Perindopril Butylamine是一种血管紧张素转化酶(ACE)抑制剂。
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ACE 抑制剂
Temocapril是一种ACE抑制剂。
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ACE 抑制剂
Cilazapril monohydrate是哒嗪血管紧张素转换酶抑制剂(ACE抑制剂),用于治疗高血压和充血性心力衰竭。
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Moexipril hydrochloride是一种有效的口服活性非巯基血管紧张素转换酶抑制剂(ACE),可作用于高血压和充血性心力衰竭。
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