CPI-613 (Devimistat)

Name: CPI-613 (Devimistat)
SKU: A11786

目录号: A11786

Dehydrogenase 抑制剂

Product Citations (2)

CPI-613 (Devimistat) Chemical Structure

CAS NO. 95809-78-2

CPI-613是合成的α-硫辛酸硫辛酸类似物的对映异构体的外消旋混合物，具有潜在的化学预防和抗肿瘤活性。

库存：现货

规格	价格	数量
5 mg	￥ 500.00
10 mg	￥ 650.00
25 mg	￥ 900.00
50 mg	￥ 1,400.00
10mM * 1mL in DMSO	￥ 500.00

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生物活性

CPI-613是合成的α-硫辛酸硫辛酸类似物的对映异构体的外消旋混合物，具有潜在的化学预防和抗肿瘤活性。

靶点信息

PDH (NCI-H460 cells)	α-ketoglutarate dehydrogenase (NCI-H460 cells)

溶解度 *

In vitro (25°C)	DMSO	74 mg/mL (190.43 mM)
	Water	Insoluble
	Ethanol	74 mg/mL (190.43 mM)
In vivo	2% DMSO+corn oil	13 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	25.73 mL	128.67 mL	257.33 mL
0.5 mM	5.15 mL	25.73 mL	51.47 mL
1 mM	2.57 mL	12.87 mL	25.73 mL
5 mM	0.51 mL	2.57 mL	5.15 mL

*The above data is based on the productmolecular weight 388.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11786
作用机制	Inhibitor (抑制剂)
M. Wt	388.6
Formula	C22H28O2S2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	95809-78-2
Synonyms	CPI613
SMILES	C1=CC=C(C=C1)CSCCC(CCCCC(=O)O)SCC2=CC=CC=C2