Immethridine hydrobromide

目录号: A13641

histamine H3 receptor 激动剂

Immethridine hydrobromide

Immethridine hydrobromide Chemical Structure

CAS NO. 87976-03-2

Immethridine hydrobromide是一种强而高选择性的组胺H3受体激动剂(pEC50 = 9.74),其选择性是H4受体的300倍(pKi值分别为9.07和6.61)。

库存: 现货

规格 价格 数量
10 mg
¥ 1,200.00
25 mg
¥ 2,500.00
50 mg
¥ 4,000.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

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Immethridine hydrobromide是一种强而高选择性的组胺H3受体激动剂(pEC50 = 9.74),其选择性是H4受体的300倍(pKi值分别为9.07和6.61)。
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 41.65 mL 208.24 mL 416.49 mL
0.5 mM 8.33 mL 41.65 mL 83.3 mL
1 mM 4.16 mL 20.82 mL 41.65 mL
5 mM 0.83 mL 4.16 mL 8.33 mL

*The above data is based on the productmolecular weight 240.103. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A13641
作用机制 Agonist (激动剂)
M. Wt 240.103
Formula C9H9N3.HBr
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 87976-03-2
Synonyms Immethridine HBr
SMILES C1=CN=CC=C1CC2=CN=CN2.Br

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