LPA Receptor

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  1. Ki16425

    Catalog No. A10501
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    LPA Receptor 拮抗剂
    ki16425是对LPA1和LPA3具有选择性的LPA受体拮抗剂,对人LPA1、LPA2和LPA3受体分别显示Ki值为0.34、6.5和0.93 μM。 了解更多
  2. Ki16198

    Catalog No. A11966
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    LPA Receptor 拮抗剂
    Ki16198是有效的LPA受体拮抗剂,可抑制LPA1和LPA3诱导的肌醇磷酸生成,Ki分别为0.34μM和0.93μM。 了解更多
  3. AM095 free base

    Catalog No. A14180
    LPA1 Receptor 拮抗剂
    AM095 free base是一种新型,有效且口服可生物利用的溶血磷脂酸1型受体(LPA1)拮抗剂,对小鼠或重组人LPA1的IC50值分别为0.73和0.98μM。 了解更多
  4. AM095

    Catalog No. A13981
    LPA1 receptor 拮抗剂
    AM095是一种有效的LPA1受体拮抗剂,因为它抑制GTPβS与过量表达重组人或小鼠LPA1的中国仓鼠卵巢(CHO)细胞膜结合,IC50值分别为0.98和0.73μM,并且没有LPA1激动作用。 了解更多
  5. AM966

    Catalog No. A13982
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    LPA1 receptor 拮抗剂
    AM966是LPA1受体(溶血磷脂酸受体)的高亲和力,选择性口服拮抗剂,IC50值为17 nM。 了解更多
  6. GRI 977143

    Catalog No. A15343
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    LPA2 激动剂
    GRI 977143是选择性溶血磷脂酸2(LPA2)受体非脂质激动剂(EC50 = 3.3 uM)。 了解更多
  7. ASP6432

    Catalog No. A18759
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    LPA1 receptor antagonist
    ASP6432 is a potent and selective Type 1 Lysophosphatidic Acid (LPA1) receptor antagonist. 了解更多
  8. AS2717638

    Catalog No. A18630
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    LPA5 antagonist
    AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF2α-, and AMPA-induced allodynia. 了解更多
  9. Radioprotectin-1

    Catalog No. A18628
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    LPA2 agonist
    Radioprotectin-1 is a potent and specific nonlipid agonist of lysophosphatidic acid receptor 2 (LPA2), with an EC50 value of 25 nM for murine LPA2 subtype. 了解更多
  10. ONO-7300243

    Catalog No. A16644
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    LPA1 antagonist
    ONO-7300243 is a novel, potent lysophosphatidic acid receptor 1 (LPA1) antagonist with IC50 of 0.16 μM. 了解更多
  11. LPA1 antagonist 1

    Catalog No. A21301
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    LPA1 antagonist
    LPA1 antagonist 1 is a highly selective Lysophosphatidic Acid receptor-1 (LPA1) antagonist with an IC50 of 25 nM. 了解更多
  12. LPA2 antagonist 1

    Catalog No. A21308
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    LPA2 antagonist
    LPA2 antagonist 1 is a LPA2 antagonist with an IC50 of 17 nM. 了解更多
  13. BMS-986020 sodium

    Catalog No. A21842
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    LPA1 antagonist
    BMS-986020 sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist. 了解更多

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