DNA Methyltransferases

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  1. Lomeguatrib

    Catalog No. A12785
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    MGMT 抑制剂
    Lomeguatrib是O6-烷基鸟嘌呤-DNA-烷基转移酶的有效抑制剂。 了解更多
  2. CM-272

    Catalog No. A17173
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    G9a/DNMT 抑制剂
    CM-272是血液恶性肿瘤中针对G9a和DNMT的可逆双重小分子抑制剂。 了解更多
  3. CM-579

    Catalog No. A18692
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    G9a/DNMT inhibitor
    CM-579 is a first-in-class reversible, dual inhibitor of G9a and DNMT, with IC50 values of 16 nM, 32 nM for G9a and DNMT, respectively. Has potent in vitro cellular activity in a wide range of cancer cells. 了解更多
  4. 6-Methyl-5-azacytidine

    Catalog No. A13391
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    DNMT inhibitor
    6-Methyl-5-azacytidine is a potent DNMT inhibitor. 了解更多
  5. O6BTG-octylglucoside

    Catalog No. A11432
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    MGMT inhibitor
    O6BTG-octylglucoside is a potent O6-methylguanine-DNAmethyl-transferase (MGMT) inhibitor, with IC50s of 32 nM in vitro (cell extracts) and 10 nM in HeLa S3 cells. 了解更多
  6. (-)-Epigallocatechin gallate

    Catalog No. A10005
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    Antioxidant, antiangiogenic, antitumor agent
    (-)-Epigallocatechin gallate是一种从绿茶中分离出来的强效抗氧化剂多酚类黄酮。 了解更多
  7. Decitabine

    Catalog No. A10292
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    DNA Methyltransferase 抑制剂
    Decitabine是一种次甲基化剂,它通过抑制DNA甲基转移酶来使DNA次甲基化。 了解更多
  8. Azacitidine(Vidaza)

    Catalog No. A10105
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    DNMT 抑制剂
    Azacitidine (Vidaza)是DNA和RNA中使用的胞嘧啶核苷的化学类似物,主要用于治疗骨髓增生异常综合症(MDS)。 了解更多
  9. SGI-110 (Guadecitabine)

    Catalog No. A12744
    DNMT 抑制剂
    SGI-110 (Guadecitabine)是第二代DNA次甲基化剂。 了解更多
  10. SGI 1027

    Catalog No. A14120
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    DNMT 抑制剂
    SGI 1027是DNMT抑制剂,对DNMT1,DNMT3A和DNMT3B的IC50分别为6、8、7.5 uM。 了解更多
  11. Procainamide HCl

    Catalog No. A14240
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    Sodium channel blocker/DNMT 抑制剂
    Procainamide HCl是钠通道阻滞剂,又是DNA甲基转移酶抑制剂。 了解更多
  12. RG108

    Catalog No. A13054
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    DNA methyltransferase 抑制剂
    RG108是DNA甲基转移酶的非核苷抑制剂,IC50为115 nM。 了解更多
  13. O6-Benzylguanine

    Catalog No. A13706
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    MGMT 抑制剂
    O6-Benzylguanine是DNA烷基转移酶的有效底物和有效灭活剂。O6-苄基鸟嘌呤是MGMT的抑制剂。 了解更多
  14. Nanaomycin A

    Catalog No. A13477
    DNMT3B 抑制剂
    Nanaomycin A是DNA甲基转移酶3B(DNMT3B)的选择性抑制剂,IC50值为500 nM。 了解更多

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