MMP

Catalog No.Inhibitor Name MMP
A12985Batimastat (BB-94)
***
A13320Ilomastat (GM6001, Galardin)
****
A14253SB-3CT
*
A12826Marimastat (BB-2516)
***
A13072NSC 405020
A10651Nobiletin

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. MMP3 inhibitor 1

    Catalog No. A13185
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    MMP-3 inhibitor
    MMP3 inhibitor 1 is a potent and highly selective MMP-3 inhibitor with an IC50 of 1 nM. 了解更多
  2. Apratastat

    Catalog No. A13330
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    dual TACE/MMPs inhibitor
    Apratastat is an orally active, potent, and reversible dual inhibitor of tumor necrosis factor-α converting enzyme (TACE) and matrix metalloproteinases (MMPs) . 了解更多
  3. T-26c

    Catalog No. A12853
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    matrix metalloproteinase-13 (MMP-13) inhibitor
    T-26c is highly potent and selective matrix metalloproteinase-13 (MMP-13) inhibitor with an IC50 of 6.75 pM and more than 2600-fold selectivity over the other related metalloenzymes. 了解更多
  4. DB04760

    Catalog No. A18548
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    MMP-13 inhibitor
    DB04760 (compound 4) is a potent, highly selective, non-zinc-chelating MMP-13 inhibitor with an IC50 of 8 nM. DB04760 significantly reduces paclitaxel neurotoxicity and has anticancer activity. 了解更多
  5. BR351

    Catalog No. A18617
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    MMP inhibitor
    BR351 is a brain penetrant MMP inhibitor with IC50s of 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13, respectively. 了解更多
  6. Doxycycline monohydrate

    Catalog No. A17813
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    MMP inhibitor
    Doxycycline monohydrate is an antibiotic and broad-spectrum metalloproteinase (MMP) inhibitor. 了解更多
  7. Doxycycline

    Catalog No. A17545
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    MMP inhibitor
    Doxycycline, an antibiotic, is an orally active and broad-spectrum metalloproteinase (MMP) inhibitor. 了解更多
  8. JNJ0966

    Catalog No. A17025
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    MMP9 抑制剂
    JNJ0966是一种高度选择性的MMP-9酶原抑制剂,IC50为440 nM。 了解更多
  9. 20(R)-Ginsenoside Rh2

    Catalog No. A15408
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    MMP 抑制剂
    20(R)-Ginsenoside Rh2是一种基质金属蛋白酶(MMP)抑制剂,可作为细胞抗增殖剂。 了解更多
  10. Batimastat sodium salt

    Catalog No. A15326
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    MMP 抑制剂
    Batimastat sodium salt是一种抗癌药物,属于称为血管生成抑制剂的药物家族。Batimastat(BB-94)是一种有效的广谱基质金属蛋白酶(MMP)抑制剂。 了解更多
  11. UK 356618

    Catalog No. A15323
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    MMP-3 抑制剂
    UK 356618是MMP-3的选择性强效抑制剂,在一系列MMP上显示出选择性。 了解更多
  12. WAY 170523

    Catalog No. A15317
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    MMP-13 抑制剂
    WAY 170523是MMP-13的选择性强效抑制剂。 了解更多
  13. UK 370106

    Catalog No. A15316
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    MMP-3/MMP-12 Inhiibitor
    UK 370106是一种高度选择性的MMP-3和MMP-12抑制剂。 了解更多
  14. Ro 32-3555

    Catalog No. A15311
    MMP 抑制剂
    Ro 32-3555是一种有效的胶原酶选择性MMP抑制剂。 了解更多
  15. PD 166793

    Catalog No. A15307
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    Broad spectrum MMP 抑制剂
    PD166793是一种细胞可渗透的化合物,可强烈抑制MMP(基质金属蛋白酶)-2,-3和-13,而弱抑制AMP脱氨酶,MMP-1,-7,-9和-14。 了解更多
  16. 4-epi-Chlortetracycline Hydrochloride

    Catalog No. A12848
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    MMP 抑制剂
    4-epi-Chlortetracycline Hydrochloride是一种四环素衍生物,可作为金属蛋白酶(MMP)抑制剂,用于治疗组织破坏性疾病和癌症。 了解更多
  17. NSC 405020

    Catalog No. A13072
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    MT1-MMP 抑制剂
    NSC-405020是一种膜1型基质金属蛋白酶(MT1-MMP)抑制剂(IC50> 100μmol/ L)。 了解更多
  18. Marimastat

    Catalog No. A12826
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    MMP 抑制剂
    Marimastat充当广谱基质金属蛋白酶抑制剂。 了解更多
  19. GM 6001

    Catalog No. A13320
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    MMP 抑制剂
    GM 6001是一种有效的,可逆的广谱抑制剂,用于含锌的蛋白酶,包括基质金属蛋白酶(MMP)。 了解更多
  20. SB-3CT

    Catalog No. A14253
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    MMP-2/MMP-9 抑制剂
    SB-3CT是一种有效的选择性明胶酶抑制剂,MMP-2和MMP-9的Ki分别为13.9 nM和600 nM。 了解更多
  21. CL-82198

    Catalog No. A13597
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    MMP-13 抑制剂
    CL-82198是人胶原酶3(也称为基质金属蛋白酶13(MMP-13))的选择性抑制剂,在10 mg/ml时产生89%的抑制作用。 了解更多
  22. ARP 100

    Catalog No. A15292
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    MMP-2 抑制剂
    ARP 100是基质金属蛋白酶2(MMP-2)的选择性抑制剂,IC50值为12 nM。 了解更多
  23. ARP 101

    Catalog No. A15293
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    MMP-2 抑制剂
    ARP 101,MMP-2的选择性抑制剂,相对于MMP-1表现出约600倍的选择性(IC50值分别为0.81和486 nM)。 了解更多
  24. CP 471474

    Catalog No. A15297
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    MMP 抑制剂
    CP 471474,广谱MMP抑制剂(对于MMP-2,MMP-13,MMP-9,MMP-3和MMP-1,IC50值分别为0.7、0.9、13、16和1170 nM)。 了解更多
  25. ONO 4817

    Catalog No. A15305
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    Broad spectrum MMP 抑制剂
    ONO 4817是广谱MMP抑制剂; MMP-12,MMP-2,MMP-8,MMP-13,MMP-9,MMP-3和MMP-7的Ki值分别为0.45、0.73、1.1、1.1、2.1、42和2500 nM,IC50 = 1600 MMP-1为nM)。 最高浓度为100μM的其他蛋白酶均无活性。 对鼠肾细胞癌的肺转移具有抗血管生成和抗侵袭特性。 了解更多
  26. TAPI-0

    Catalog No. A13724
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    TACE/MMP 抑制剂
    TAPI-0是TACE(IC50 = 50-100 nM)以及其他基质和膜金属蛋白酶的抑制剂。 了解更多
  27. Abametapir

    Catalog No. A15945
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    metalloproteinase 抑制剂
    ABAMETAPIR是Xeglyze乳液的活性成分。ABAMETAPIR抑制金属蛋白酶;对卵子发育,若虫和成年虱子存活至关重要的生理过程必不可少的酶。 了解更多
  28. Doxycycline HCl

    Catalog No. A10745
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    Doxycycline Hydrochloride是具有类似抗菌活性的合成四环素衍生物。 了解更多
  29. DC_AC50

    Catalog No. A16043
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    Atox1/CCS 抑制剂
    DC_AC50是铜转运蛋白Atox1和CCS的抑制剂,导致细胞铜转运的中断。 了解更多
  30. TAPI-2

    Catalog No. A14009
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    TACE/MMP 抑制剂
    TAPI-2是TACE,ADAM,ACE分泌酶和其他MMP(金属蛋白酶)的抑制剂。TAPI-2阻止DCC7,APP,TNFα,L-选择素,NOTCH,TGFα,IL-6R9,erbB2/HER2和ACE的释放。该抑制剂已用于组织培养。 了解更多
  31. TMI-1

    Catalog No. A17212
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    TACE/MMP 抑制剂
    TMI-1是ADAM17(TACE)和MMP的新型活性双重抑制剂。 了解更多
    • 最新产品

    Incyclinide

    Catalog No. A17240
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    MMP inhibitor
    Iincyclinide, also known as CMT-3 and COL-3, is a MMP inhibitor and a chemically-modified tetracycline with potential antineoplastic activity. Incyclinide inhibits matrix metalloproteinases (MMPs), thereby inducing extracellular matrix degradation, and inhibiting angiogenesis, tumor growth and invasion, and metastasis. This agent also causes mitochondrial depolarization in tumor cells and induces both cellular apoptosis and tissue necrosis. 了解更多
  32. TAPI-1

    Catalog No. A14070
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    TACE/MMP 抑制剂
    TAPI-1是一种ADAM17/TACE抑制剂, 其对细胞因子受体有抑制作用。 了解更多
  33. Batimastat (BB-94)

    Catalog No. A12985
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    MMP 抑制剂
    Batimastat (BB-94)是多种基质金属蛋白酶(MMP)的强效合成抑制剂,包括间质胶原酶(IC50 = 3 nM),溶血素(IC50 = 20 nM),Mr 72,000型IV胶原酶(IC50 = 4) nM),92,000型IV胶原酶先生(IC50 = 4 nM)和基质溶素(IC50 = 6 nM)。它是一种低分子量(MW = 478)的肽样胶原蛋白底物类似物,由类似物结合而成,分别与MMP和催化活性锌原子结合在一起。 了解更多
  34. CTS-1027

    Catalog No. A11345
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    Matrix Metalloproteinase 抑制剂
    CTS-1027是一种有效的MMP抑制剂,可预防TNFα和α-Fas诱导的肝损伤。 了解更多

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