“raf”的搜索结果

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  1. ERK-IN-1

    Catalog No. A19080
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    RAF/ERK1/2 inhibitor
    ERK-IN-1 (compound B) is a RAF and ERK1/2 inhibitor in the treatment of a proliferative disease characterized by activating mutations in the MAPK pathway. 了解更多
  2. LY3214996

    Catalog No. A16843
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    ERK 抑制剂
    LY3214996是一种选择性的新型ERK1/2抑制剂,在生化分析中两种酶的IC50为5 nM。它有效抑制BRAF和RAS突变癌细胞系中的细胞磷酸RSK1。 了解更多
  3. APS-2-79

    Catalog No. A16231
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    KSR/Ras 抑制剂
    APS-2-79是RAF通过直接结合KSR活性位点而使MEK磷酸化的拮抗剂。 了解更多

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