“angiotensin converting enzyme ace”的搜索结果

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  1. Sparsentan

    Catalog No. A20879
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    angiotensin II and endothelin A receptor antagonist
    Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多
  2. NS-2028

    Catalog No. A21643
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    sGC inhibitor
    NS-2028 is a highly selective soluble Guanylyl Cyclase (sGC) inhibitor with IC50 values of 30 nM and 200 nM for basal and NO-stimulated enzyme activity. 了解更多
  3. Olinciguat

    Catalog No. A13670
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    guanylate cyclase (sGC) stimulator
    Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator with concentration-dependent stimulation of sGC in purified rat and human enzyme assays and a whole cell assay. 了解更多
  4. Mavoglurant racemate

    Catalog No. A21799
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    mGlu5 receptor antagonist
    Mavoglurant (racemate) is the racemate of mavoglurant. Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. 了解更多
  5. Taranabant racemate

    Catalog No. A21699
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    CB1 antagonist/inverse agonist
    Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor extracted from patent WO 2004048317 A1. 了解更多
  6. (±)-Ibipinabant

    Catalog No. A21439
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    CB-1 receptor antagonist
    (±)-Ibipinabant ((±)-SLV319) is the racemate of SLV319. (±)-Ibipinabant ((±)-SLV319) is a potent and selective cannabinoid-1 (CB-1) receptor antagonist with an IC50 of 22 nM. 了解更多
  7. Pexacerfont

    Catalog No. A14105
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    CRF1 receptor antagonist
    Pexacerfont is a selective corticotropin-releasing factor (CRF1) receptor antagonist with IC50 of 6.1??0.6 nM for human CRF1 receptor. 了解更多
  8. Kynurenic acid sodium

    Catalog No. A20000
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    GPR35/CXCR8 agonist
    Kynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. 了解更多
  9. CAY10471 Racemate

    Catalog No. A11760
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    Prostaglandin D2 receptor CRTH2 antagonist
    CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多
  10. MHP 133

    Catalog No. A20058
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    AChE /M1/M2/5HT4/I2 inhibitor
    MHP 133 is a drug with multiple CNS targets, and inhibits acetylcholinesterase (AChE) with Ki of 69 μM; also active against muscarinic M1 and M2 receptors, serotonin 5HT4 receptors, and imidazole I2 receptors. 了解更多
  11. Kynurenic acid

    Catalog No. A16581
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    GPR35/CXCR8 拮抗剂
    Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多
  12. Anisodamine

    Catalog No. A18215
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    alpha-1 adrenergic receptors / mAChRs inhibitor
    Anisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多
  13. Benorylate

    Catalog No. A17501
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    Prostaglandin Receptor inhibitor
    Benorilate, also known as Win-11450, is an ester of aspirin and paracetamol with analgesic, antipyretic, and anti-inflammatory activity used in the treatment of rheumatoid diseases. Benorilate has less severe side effects than aspirin. 了解更多
  14. Melitracen hydrochloride

    Catalog No. A17494
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    dopamine D1/2 receptor antagonist
    Melitracen HCl ia potential dopamine D1/2 receptor antagonist used to treat depression. It is often co-administered with flupenthixol as a treatment for trigeminal neuralgia. It does not effect cardiovascular function. 了解更多
  15. LY 344864 racemate

    Catalog No. A17015
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    5-HT1F receptor 激动剂
    LY 344864 racemate是5-HT1F受体激动剂。 了解更多
  16. Theophylline-7-acetic acid

    Catalog No. A16822
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    Adenosine receptor 拮抗剂
    Theophylline-7-acetic acid是腺苷受体拮抗剂,是黄嘌呤类化学物质的兴奋剂。 了解更多
  17. Acebutolol HCl

    Catalog No. A16387
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    β-adrenergic receptors 拮抗剂
    Acebutolol HCl是一种β-肾上腺素能受体拮抗剂,用于治疗高血压,心绞痛和心律不齐。 了解更多
  18. Phenylpiracetam

    Catalog No. A15211
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    Dopamine reuptake 抑制剂
    Phenylpiracetam是促智药物吡乙酰胺的苯基化衍生物。它被用作促智药物,效力比吡乙酰胺高30-60倍。 了解更多
  19. Guanabenz acetate

    Catalog No. A13635
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    2A-AR adrenergic 激动剂
    Guanabenz acetate是a2A-AR肾上腺素能激动剂和IGRS(咪唑啉I2结合位点)选择性配体。 了解更多
  20. Lixisenatide

    Catalog No. A14076
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    GLP-1 receptor 激动剂
    Lixisenatide抑制胰高血糖素释放,显着降低餐后胰高血糖素。对糖尿病(T2DM)有促进作用。 了解更多
  21. Parathyroid Hormone 1-34, Human

    Catalog No. A12790
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    Parathyroid Hormone 1-34, Human包含hPTH的34个N端残基。 甲状旁腺1(PTH1)和甲状旁腺2(PTH2)受体的激动剂,其在 HEK293 细胞中的 IC50 值为 2 nM。 了解更多
  22. Octreotide Acetate

    Catalog No. A12782
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    somatostatin receptor 拮抗剂
    Octreotide是sst2,sst3和sst5生长抑素受体的肽激动剂。克隆的人类生长抑素受体的IC50/Kd值(nM)为:290-1140(sst1),0.4-2.1(sst2),4.4-34.5(sst3),> 1000(sst4)和5.6-32(sst5)。 了解更多
  23. Roxatidine acetate hydrochloride

    Catalog No. A11921
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    Roxatidine acetate hydrochloride是一种用于溃疡治疗的组胺H2受体拮抗剂。 了解更多

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