“jwh 370”的搜索结果

产品 151 到 161 共 161个

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  1. PS210

    Catalog No. A22109
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    protein kinase PDK1 inhibitor
    PS210 is a substrate-selective protein kinase PDK1 inhibitor that acts by binding to the PIF-pocket allosteric docking site. 了解更多
  2. RY785

    Catalog No. A22104
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    inhibitor of Kv2.1 and Kv2.2
    RY785 (Kv2-IN-A1) is an inhibitor of Kv2.1 and Kv2.2. 了解更多
  3. Avelumab

    Catalog No. A18234
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    PD-1/PD-L1
    Avelumab is a fully human IgG1 anti-PD-L1 monoclonal antibody with potential antibody-dependent cell-mediated cytotoxicity. 了解更多
  4. Mosapride citrate

    Catalog No. A10607
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    5-HT4-receptor 激动剂
    Mosapride citrate起5-HT4受体激动剂和5-HT3受体拮抗剂的作用。 了解更多
  5. KN-92

    Catalog No. A15137
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    CaMK-II 抑制剂
    KN-92是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II(CaMKII)的选择性抑制剂,竞争性阻断CaM与激酶的结合(Ki = 370 nM)。 了解更多
  6. KN-92 phosphate

    Catalog No. A15139
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    CaMKII 抑制剂
    KN-92 phosphate是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II(CaMKII)的选择性抑制剂,竞争性阻断CaM与激酶的结合(Ki = 370 nM)。 了解更多
  7. FCCP

    Catalog No. A16545
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    ionophore
    FCCP是一种离子载体,是一种可移动的离子载体。它是线粒体中氧化磷酸化的有效解偶联剂,可通过跨细胞膜转运质子来破坏ATP合成。 了解更多
  8. (-)-Ibuprofenamide

    Catalog No. A19398
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    (-)-Ibuprofenamide is an amide prodrug of Ibuprofen with anti-inflammatory activity. Ibuprofen is an anti-inflammatory inhibitor targeting COX-1 and COX-2 with IC50s of 13 μM and 370 μM, respectively. 了解更多
  9. NSC 191412

    Catalog No. A22657
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    NSC 191412 (1-(4-Fluorophenyl)-3-phenylthiourea) is an active compound. 了解更多
  10. NSC 80538

    Catalog No. A22655
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    NSC 80538 (1-(4-Chlorophenyl)-3-(4-fluorophenyl)thiourea) is an inhibitor of MEK Kinase PB1 Domains in Multiplex HTS Assay. 了解更多
  11. KN-93 phosphate

    Catalog No. A22229
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    membrane-permeant synthetic inhibitor
    KN-93 phosphate is a novel membrane-permeant synthetic inhibitor of purified neuronal CaMK-II, with Ki of 370 nM. 了解更多

产品 151 到 161 共 161个

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