Histamine Receptors

产品 1 到 50 共 62个

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  1. Decloxizine

    Catalog No. A20964
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    histamine 1 receptor antagonist
    Decloxizine(UCB-1402; NSC289116) is a histamine 1 receptor antagonist. 了解更多
  2. GSK189254A

    Catalog No. A22005
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    histamine H3 receptor antagonist
    GSK189254A (GSK189254) is a novel, potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively. 了解更多
  3. Niperotidine

    Catalog No. A21981
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    histamine H2-receptor antagonist
    Niperotidine is a histamine H2-receptor antagonist. 了解更多
  4. JNJ-5207852

    Catalog No. A21480
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    histamine H3 receptor antagonist
    JNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively. 了解更多
  5. PF-03654746 Tosylate

    Catalog No. A21434
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    histamine H3 receptor antagonist
    PF-03654746 Tosylate is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多
  6. PF-03654746

    Catalog No. A21429
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    histamine H3 receptor antagonist
    PF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多
  7. Toreforant

    Catalog No. A21058
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    histamine H4 receptor (H4R) antagonist
    Toreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多
  8. Chlorcyclizine hydrochloride

    Catalog No. A18025
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    histamine H1 antagonist
    Chlorcyclizine hydrochloride is a histamine H1 antagonist. 了解更多
  9. H4 Receptor antagonist 1

    Catalog No. A18929
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    histamine H4 receptor inverse agonist
    H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. 了解更多
  10. Buclizine HCl

    Catalog No. A15666
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    Buclizine hydrochloride是哌嗪衍生物家族的抗组胺药和抗胆碱能药。 了解更多
  11. Cyproheptadine hydrochloride

    Catalog No. A16169
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    serotonin/histamine2 拮抗剂
    Cyproheptadine hydrochloride是抗组胺药,是5-羟色胺和组胺的拮抗剂。 了解更多
  12. Lidocaine hydrochloride

    Catalog No. A16132
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    Histamine H1-receptor 激动剂
    Lidocaine hydrochloride是用作抗心律不齐药物的局部麻醉药和心脏抑制剂。 了解更多
  13. CarbinoxaMine Maleate

    Catalog No. A16129
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    histamine-H1 receptor blocking agent
    Carbinoxamine maleate是一种具有抗组胺和抗胆碱能特性的组胺-H1受体阻断剂。 了解更多
  14. Bavisant dihydrochloride hydrate

    Catalog No. A15016
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    H3 receptor 拮抗剂
    Bavisant dihydrochloride hydrate是人类H3受体的高度选择性口服活性拮抗剂。 了解更多
  15. Bavisant dihydrochloride

    Catalog No. A15015
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    H3 receptor 拮抗剂
    Bavisant dihydrochloride是一种人类H3受体的高选择性,口服活性拮抗剂。 了解更多
  16. Zaltidine

    Catalog No. A15285
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    H2-receptor 拮抗剂
    Zaltidine是H2受体拮抗剂,具有抗分泌作用。 了解更多
  17. Pitolisant oxalate

    Catalog No. A15214
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    Nonimidazole inverse 激动剂
    Pitolisant oxalate是一种在重组人H3受体上的新型,有效且选择性的壬咪唑反向激动剂(Ki = 0.16 nM)。 了解更多
  18. Pitolisant hydrochloride

    Catalog No. A15213
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    Nonimidazole inverse 激动剂
    Pitolisant hydrochloride是一种在重组人H3受体(Ki = 0.16 nM)处新颖,有效且选择性的壬二唑反向激动剂。 了解更多
  19. Ebrotidine

    Catalog No. A15075
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    H2-receptor 拮抗剂
    Ebrotidine是一种竞争性的H2受体拮抗剂(Ki = 127.5 nM),具有有效的抗分泌活性和胃保护作用。 了解更多
  20. Clemizole hydrochloride

    Catalog No. A15047
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    H1 histamine receptor 拮抗剂
    Clemizole hydrochloride是H1组胺受体的拮抗剂,对NS4B RNA结合的IC50值为8 mM。 了解更多
  21. Alcaftadine

    Catalog No. A16393
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    H1 histamine receptor 拮抗剂
    Alcaftadine是H1受体的高亲和力配体,其pKi(8.5)与其他H1抗组胺药相当。Alcaftadine还是H2和H4受体的拮抗剂,对H3受体没有亲和力。 了解更多
  22. Antazoline HCl

    Catalog No. A16411
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    Histamine H1 receptor 抑制剂
    Antazoline HCl是第一代抗组胺药,可与组胺H1受体结合并阻断内源性组胺的作用。 了解更多
  23. Azatadine dimaleate

    Catalog No. A16418
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    Histamine/cholinergic 抑制剂
    Azatadine是一种组胺和胆碱能抑制剂,IC50分别为6.5 nM和10 nM。 了解更多
  24. Cyclizine 2HCl

    Catalog No. A16472
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    Histamine H1 receptor 拮抗剂
    Cyclizine 2HCl是具有组胺H1受体拮抗剂活性的哌嗪衍生物。 了解更多
  25. Terfenadine

    Catalog No. A17373
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    H1 histamine receptor antagonist
    Terfenadine ((??)-Terfenadine) is a potent open-channel blocker of hERG with an IC50 of 204 nM. Terfenadine, an H1 histamine receptor antagonist, acts as a potent apoptosis inducer in melanoma cells through modulation of Ca2+ homeostasis. Terfenadine induces ROS-dependent apoptosis, simultaneously activates Caspase-4, -2, -9 and induces p73, Noxa. 了解更多
  26. Levocetirizine Dihydrochloride

    Catalog No. A17440
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    L-isomer of cetirizine and histamine H1 receptor antagonist
    Levocetirizine dihydrochloride is a L-isomer of cetirizine and histamine H1 receptor antagonist. It incrases levels of CD4+ CD25+ T cells and decreases levels of eosinophils, decreasing allergy symptoms. 了解更多
  27. Hydroxyzine pamoate

    Catalog No. A17712
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    Histamine H1 receptor antagonist
    Hydroxyzine pamoate is an histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIRIZINE, it does cause drowsiness. 了解更多
  28. Diphenylpyraline hydrochloride

    Catalog No. A17717
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    antihistamine
    Diphenylpyraline hydrochloride is a first-generation antihistamine with anticholinergic effects of the diphenylpiperidine class. 了解更多
  29. Acrivastine

    Catalog No. A17746
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    Histamine 1 receptor antagonist
    Acrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis. 了解更多
  30. Mebhydrolin napadisylate

    Catalog No. A17997
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    histamine H1-receptor antagonist
    Diazoline is a histamine H1-receptor antagonist. 了解更多
  31. Mequitazine

    Catalog No. A18206
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    Histamine H1 antagonist
    Mequitazine is a potent histamine H1 antagonist or antihistamine. It competes with histamine for the normal H1-receptor sites on effector cells of the gastrointestinal tract, blood vessels and respiratory tract. 了解更多
  32. Ciproxifan maleate

    Catalog No. A11117
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    H3-receptor 拮抗剂
    Ciproxifan maleate是一种有效的选择性H3组胺受体拮抗剂。 了解更多
  33. Azelastine HCl (Allergodil)

    Catalog No. A10117
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    Azelastine HCl (Allergodil)是有效的第二代选择性组胺拮抗剂(组胺-H1-受体拮抗剂)。 了解更多
  34. Brompheniramine

    Catalog No. A11699
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    Brompheniramine是一种组胺H1受体拮抗剂。 了解更多
  35. Clemastine fumarate

    Catalog No. A10226
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    Histamine Receptor antagonis
    Clemastine fumarate是一种选择性的组胺H1拮抗剂。它与组胺H1受体结合,从而阻断了内源性组胺的作用,从而暂时缓解了由组胺引起的阴性症状。 了解更多
  36. Ciproxifan

    Catalog No. A11360
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    Ciproxifan是一种非常有效的组胺H3反向激动剂/拮抗剂。 了解更多
  37. Cyproheptadine hydrochloride

    Catalog No. A11709
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    Cyproheptadine hydrochloride 是 5-HT2 受体拮抗剂,IC50为0.6 nM。 了解更多
  38. Orphenadrine citrate

    Catalog No. A11712
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    NMDA receptor 拮抗剂
    Orphenadrine柠檬酸盐是NMDA受体拮抗剂,Ki为6.0μM,还是HERG钾离子通道阻断剂。 了解更多
  39. Lafutidine

    Catalog No. A11714
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    H2 receptor 拮抗剂
    Lafutidine是具有多峰作用机制的第二代H2受体拮抗剂。 了解更多
  40. Mizolastine

    Catalog No. A11724
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    Mizolastine是组胺H1受体拮抗剂,IC50为47 nM。 了解更多
  41. Asenapine maleate

    Catalog No. A10091
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    H1 拮抗剂
    Asenapine maleate平对多种受体具有高亲和力(pKi),包括5-羟色胺5-HT1A(8.6),5-HT1B(8.4),5-HT2A(10.2),5-HT2B(9.8),5-HT2C(10.5),5 -HT5A(8.8),5-HT6(9.5)和5-HT7(9.9)受体,肾上腺素α1(8.9),α2A(8.9),α2B(9.5)和α2C(8.9)受体,多巴胺D1( 8.9),D2(8.9),D3(9.4)和D4(9.0)受体以及组胺H1(9.0)和H2(8.2)受体。 了解更多
  42. Cetirizine Dihydrochloride

    Catalog No. A10195
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    Cetirizine Dihydrochloride是第二代抗组胺药,是羟嗪的主要代谢产物,是用于治疗过敏,花粉症,血管性水肿和荨麻疹的消旋选择性H1受体反向激动剂。 了解更多
  43. Chlorpheniramine maleate

    Catalog No. A10205
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    Chlorpheniramine maleate是用于预防过敏性疾病如鼻炎和荨麻疹症状的第一代烷基胺抗组胺药。 了解更多
  44. Cimetidine

    Catalog No. A10218
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    H2-receptor 拮抗剂
    Cimetidine是一种抑制胃酸产生的组胺H2受体拮抗剂。 了解更多
  45. Bepotastine Besilate

    Catalog No. A11340
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    Histamine Receptor 拮抗剂
    Bepotastine Besilate是组胺H1受体激动剂。 了解更多
  46. Roxatidine acetate hydrochloride

    Catalog No. A11921
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    Roxatidine acetate hydrochloride是一种用于溃疡治疗的组胺H2受体拮抗剂。 了解更多
  47. Rupatadine Fumarate

    Catalog No. A12356
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    PAFR 抑制剂/H1 receptor 抑制剂
    Rupatadine Fumarate是PAFR和组胺(H1)受体的抑制剂,Ki分别为550和102 nM。 了解更多
  48. Rupatadine

    Catalog No. A11222
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    PAFR 抑制剂/H1 receptor 抑制剂
    Rupatadine是PAFR和组胺(H1)受体的抑制剂,Ki分别为550和102 nM。 了解更多
  49. Loratadine

    Catalog No. A10538
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    Loratadine是一种非镇静抗组胺药,抑制组胺诱导的内皮细胞分泌IL-6和IL-8的活性。氯雷他定是一种选择性外周组胺h1受体拮抗剂,IC50 > 32 μM。 了解更多
  50. Fexofenadine HCl

    Catalog No. A11859
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    COX 抑制剂/histamine H1 receptor 激动剂
    Fexofenadine Hydrochloride是一种抗组胺药,可抑制Cox-1,Cox-2,并且是组胺H1受体激动剂,IC50为246 nM。 了解更多

产品 1 到 50 共 62个

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