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GPR35/CXCR8 agonist
Kynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8.
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GPR35/CXCR8 拮抗剂
Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8.
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5-HT1F receptor 激动剂
LY 344864 racemate是5-HT1F受体激动剂。
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2A-AR adrenergic 激动剂
Guanabenz acetate是a2A-AR肾上腺素能激动剂和IGRS(咪唑啉I2结合位点)选择性配体。
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GLP-1 receptor 激动剂
Lixisenatide抑制胰高血糖素释放,显着降低餐后胰高血糖素。对糖尿病(T2DM)有促进作用。
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