“betaine hydrochloride”的搜索结果
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β1-selective adrenergic receptor agonist
Norepinephrine hydrochloride (Levarterenol hydrochloride; L-Noradrenaline hydrochloride) is a β1-selective adrenergic receptor agonist with EC50 of 5.37 μM.
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beta-adrenergic agonist
Nylidrin hydrochloride is a beta-adrenergic agonist. Nylidrin hydrochloride is shown to be an effective inhibitor of IgE-mediated release of histamine from human basophils, and thus can be used as antiallergic agent.
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Adrenergic alpha-1 agonist
Midodrine hydrochloride is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of hypotension. It improves clinical outcome of chronic hypotension.
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alpha-1 adrenergic agonist
Methoxamine Hydrochloride is an alpha-1 adrenergic agonist that causes prolonged peripheral vasoconstriction.
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β2-adrenergic receptor agonist
Tulobuterol Hydrochloride is a long-acting beta2-adrenergic receptor agonist.
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α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂
Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。
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Alpha adrenergic 激动剂
Clonidine hydrochloride被归类为中枢作用的α肾上腺素能激动剂。Clonidine主要作为咪唑啉受体激动剂。
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Adrenergic Receptor 激动剂
Detomidine hydrochloride是具有镇痛作用的镇静剂。α2-肾上腺素能激动剂产生剂量依赖性的镇静和镇痛作用,并通过激活α2儿茶酚胺受体介导,从而引起负反馈反应,从而减少兴奋性神经递质的产生。
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adrenergic alpha-2 receptor 激动剂
Medetomidine Hydrochloride是一种肾上腺素α2-受体激动剂,Ki为1.08 nM,比作用于α1-adrenoceptor选择性高1620倍。由于其镇痛和镇静作用而被用于兽医学。
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Adrenergic Receptor 激动剂
Tetrahydrozoline Hydrochloride是一种引起结膜血管收缩的α激动剂。
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beta-Adrenergic agonist
Ractopamine HCl is a beta-Adrenergic agonist. It acts by being a full agonist at the TAAR1.
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Adrenergic Receptor 激动剂
Xylazine hydrochloride是α2A-AR、α2B-AR和α2C-AR的活化剂。
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alpha2-adrenoceptor 激动剂
Dexmedetomidine hydrochloride是美托咪啶的活性异构体,它充当有效的,高度选择性的α2-AR(α2-肾上腺素受体)激动剂。
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α2A-adrenoceptor 激动剂
Guanfacine hydrochloride是一种抗高血压药,是一种选择性的α2A肾上腺素受体激动剂,Kd为31 nM,选择性是α2B肾上腺素受体的60倍。
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α1-adrenergic receptor 激动剂
Phenylephrine HCl是一种选择性的α1肾上腺素能受体激动剂,主要用作减充血剂,扩张瞳孔和增加血压的药物。
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alpha-1 adrenergic 激动剂
Oxymetazoline是一种选择性的α-1激动剂和部分α-2激动剂局部减充血剂,以盐酸羟甲唑啉的形式使用。
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Adrenoceptors 激动剂
Dobutamine hydrochloride是一种直接作用剂,其主要活性来自刺激心脏的β1肾上腺素能受体,增加收缩力和心输出量。
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