主页 /
搜索结果：“glucagon receptor”

“glucagon receptor”的搜索结果

Quick View
L-APB

Catalog No. A21872
Quick View

添加到收藏
mGluRs M3 agonist

L-APB is a potent and specific agonist for the group III mGluRs, with EC50s of 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6 and mGlu7 receptors, respectively. 了解更多

Bulk Inquiry
Quick View
O-Phospho-L-serine

Catalog No. A21159
Quick View

添加到收藏
group III mGluR receptors agonist

O-Phospho-L-serine is the immediate precursor to L-serine in the serine synthesis pathway, and an agonist at the group III mGluR receptors (mGluR4, mGluR6, mGluR7, and mGluR8); O-Phospho-L-serine also acts as a weak antagonist for mGluR1 and a potent antagonist for mGluR2. 了解更多

Bulk Inquiry
Quick View
Eglumegad

Catalog No. A21005
Quick View

添加到收藏
group II (mGlu2/3) receptor agonist

Eglumegad (LY354740) is a highly potent and selective group II (mGlu2/3) receptor agonist with IC50s of 5 and 24 nM on transfected human mGlu2 and mGlu3 receptors, respectively. 了解更多

Bulk Inquiry
Quick View
LY2812223

Catalog No. A21100
Quick View

添加到收藏
mGlu2 receptor agonist

LY2812223 is a highly potent, functionally selective mGlu2 receptor agonist with mGlu2 binding affinity for mGlu2 and mGlu3 (Ki=144 nM and 156 nM, respectively). 了解更多

Bulk Inquiry
Quick View
LY2794193

Catalog No. A19131
Quick View

添加到收藏
mGlu3 receptor agonist

LY2794193 is a highly potent and selective mGlu3 receptor agonist (hmGlu3 Ki=0.927 nM??EC50=0.47 nM; hmGlu2 Ki=412 nM??EC50=47.5 nM). 了解更多

Bulk Inquiry
Quick View
VU6005649

Catalog No. A17023
Quick View

添加到收藏
CNS penetrant mGlu7/8 receptor 激动剂

VU6005649是一种CNS渗透性mGlu7/8受体激动剂，对mGlu7受体和mGlu8受体的EC50分别为0.65 μM和2.6 μM。了解更多

Bulk Inquiry
Quick View
Kainic acid monohydrate

Catalog No. A13485
Quick View

添加到收藏
Kainate receptor 激动剂

Kainic acid monohydrate是海藻酸酯类离子型谷氨酸受体激动剂。可在体内诱发癫痫发作和神经退行性变，也已用于在啮齿动物中诱发实验性癫痫和检查兴奋性诱发的神经元凋亡机制。了解更多

Bulk Inquiry
Quick View
Ibotenic Acid

Catalog No. A14006
Quick View

添加到收藏
NMDA& mGlu receptor 激动剂

Ibotenic Acid是最初从鹅膏菌属物种中分离出来的一种神经兴奋性氨基酸，它起着NMDA和代谢型谷氨酸受体激动剂的作用。了解更多

Bulk Inquiry
Quick View
LY 379268

Catalog No. A13123
添加到收藏
mGlu2 receptor 激动剂

LY 379268是高选择性的II类mGlu受体激动剂（对于hmGlu2和hmGlu3而言，EC50值分别为2.69和4.48 nM），其选择性是I类和III类受体的80倍以上。了解更多

Bulk Inquiry