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  1. TAK-960 hydrochloride

    Catalog No. A21703
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    PLK1 inhibitor
    TAK-960 hydrochloride is an orally available, selective inhibitor of polo-like kinase 1 (PLK1), with an IC50 of 0.8 nM at 10 μM ATP; TAK-960 hydrochloride also shows inhibitory activities against PLK2 and PLK3, with IC50s of 16.9 and 50.2 nM, respectively. 了解更多
  2. TAK-901

    Catalog No. A11067
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    Aurora Kinase A/B 抑制剂
    TAK-901是一种新型Aurora A/B抑制剂,IC50为21 nM/15 nM。它不是细胞JAK2,c-Src或Abl的有效抑制剂。 了解更多
  3. TAK-960

    Catalog No. A11146
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    PLK1 抑制剂?
    TAK-960是新型的,口服可用的polo样激酶1选择性抑制剂,具有广谱的临床前抗肿瘤活性。 了解更多

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