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Letaxaban (TAK-442)
Catalog No. A12871 factor Xa 抑制剂Letaxaban (TAK-442)是一种有效的，选择性的，口服活性的Xa抑制剂，是一种四氢嘧啶-2（1H）-衍生物。TAK-442在贫血小板的人[半最大抑制浓度（IC（50））：53 nM，TAK-442]和大鼠（IC（50）：32 nM，TAK-442）血浆中抑制内源性FXa活性。 了解更多 -
TAK-242 S enantiomer
Catalog No. A15253 TLR4 抑制剂TAK-242的S对映体。TAK-242（Resatorvid），Toll样受体（TLR）4信号转导的小分子抑制剂。TAK-242用于治疗败血症和败血性休克。 了解更多 -
TAK-700 Salt (Orteronel Salt)
Catalog No. A13515 CYP17A1/androgen synthesis 抑制剂TAK-700 Salt (Orteronel Salt)是一种雄激素合成抑制剂。它选择性地抑制在睾丸，肾上腺和前列腺肿瘤组织中表达的酶CYP17A。 了解更多 -
TAK-220
Catalog No. A20618 -
TAK-960 hydrochloride
Catalog No. A21703 PLK1 inhibitorTAK-960 hydrochloride is an orally available, selective inhibitor of polo-like kinase 1 (PLK1), with an IC50 of 0.8 nM at 10 μM ATP; TAK-960 hydrochloride also shows inhibitory activities against PLK2 and PLK3, with IC50s of 16.9 and 50.2 nM, respectively. 了解更多 -
TAK-438 (vonoprazan)
Catalog No. A11239 -
TAK-659 hydrochloride
Catalog No. A21885 Syk inhibitorTAK-659 hydrochloride is a potent, selective and orally available spleen tyrosine kinase (Syk) inhibitor with an IC50 of 3.2 nM. 了解更多 -
TAK-063
Catalog No. A15799 -
TAK-779
Catalog No. A13846 -
TAK-441
Catalog No. A11351 -
TAK-960
Catalog No. A11146 -
TAK-700 (Orteronel)
Catalog No. A11044 -
Mubritinib (TAK 165)
Catalog No. A10612 HER2/ErbB2 抑制剂Mubritinib (TAK 165)是一种有效的EGFR和p34cdc2抑制剂，IC50分别为6 nM和0.2 ?M。Mubritinib（TAK 165）也抑制p33cdk2和p33cdk5。 了解更多 -
(R)-Simurosertib
Catalog No. A21894 CDC7 kinase inhibitor(R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib, Simurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. 了解更多 -
Relugolix
Catalog No. A17783 GnRH antagonistRelugolix is a novel, non-peptide, orally active gonadotropin-releasing hormone (GnRH) antagonist with IC50 of 0.33 nM in the presence of 40% fetal bovine serum, TAK-385 possesses higher affinity and potent antagonistic activity compared with TAK-013. 了解更多 -
Ramelteon (TAK-375)
Catalog No. A10777 MT1/MT2-Receptor 激动剂Ramelteon (TAK-375)是melatonin受体激动剂，对褪黑激素MT1（IC50 = 28.5±8.55 pM）和MT2（20.1±9.25 pM）受体均具有高亲和力，并且相对于MT3受体具有选择性。 了解更多 -
Soticlestat
Catalog No. A22516 Soticlestat, also known as TAK 935 and OV935, is an inhibitor of the enzyme cholesterol 24-hydroxylase (CH24H). 了解更多 -
Sipoglitazar
Catalog No. A22625 PPARγ agonistSipoglitazar, also known as TAK-654, is a PPARγ agonist potentially for the treatment of diabetes. 了解更多 -
Simurosertib
Catalog No. A20392 CDC7 inhibitorSimurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. 了解更多 -
Vonoprazan free base
Catalog No. A18007 potassium-competitive acid blockerVonoprazan (TAK-438 free base) is an orally active potassium-competitive acid blocker which inhibits H+, K+-ATPase activity with an IC50 of 19 nM. 了解更多 -
Lapaquistat acetate
Catalog No. A20851 squalene synthase inhibitorLapaquistat acetate (TAK-475) is a squalene synthase inhibitor, blocking the conversion of farnesyl diphosphate (FPP) to squalene. 了解更多 -
Azilsartan (TAK-536)
Catalog No. A11775 -
Mobocertinib
Catalog No. A22334 inhibitor of EGFR and HER2 oncogenic mutantsMobocertinib (TAK-788) is a potent and orally active inhibitor of EGFR and HER2 oncogenic mutants, including exon 20 insertions, with selectivity over WT EGFR. Antitumor activity. 了解更多 -
Mobocertinib succinate
Catalog No. A22240 EGFR/HER2 oncogenic mutants inhibitorMobocertinib succinate (TAK-788 succinate) is a potent and orally active inhibitor of EGFR and HER2 oncogenic mutants, including exon 20 insertions, with selectivity over WT EGFR. Antitumor activity. 了解更多 -
Orteronel (racemic)
Catalog No. A22508 Orteronel (racemic) is a mixture of S-Orteronel and R-Orteronel isomers. 了解更多 -
Imiglitazar
Catalog No. A20080 PPARα/ PPARγ1 agonistImiglitazar (TAK559) is a potent and dual human PPARα and PPARγ1 agonist with EC50 values of 67 and 31 nM. 了解更多 -
Azilsartan D5
Catalog No. A21600 angiotensin II type 1 receptor antagonistAzilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. 了解更多 -
Azilsartan medoxomil monopotassium
Catalog No. A20860 angiotensin II receptor type 1 antagonistAzilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多 -
Resatorvid
Catalog No. A11543 TLR4 inhibitorResatorvid (TAK-242) is a selective Toll-like receptor 4 (TLR4) inhibitor and plays pivotal role in various inflammatory diseases. 了解更多 -
Bamirastine
Catalog No. A13325 Bamirastine inhibits ligand binding to recombinant human histamine H1 receptors (rhH1R) with an IC50 value of 17.3 nM. 了解更多 -
Cenicriviroc Mesylate
Catalog No. A17028 CCR2/5 receptors 抑制剂Cenicriviroc(TAK-652,TBR-652)是CCR2和CCR5受体的抑制剂，可使其充当防止病毒进入人细胞的进入抑制剂 了解更多 -
Azilsartan Medoxomil
Catalog No. A16420 angiotensin II receptor type 1 拮抗剂Azilsartan medoxomil是一种口服给药的1型血管紧张素II受体拮抗剂，IC50为0.62 nM。 了解更多 -
MLN1117 (Serabelisib)
Catalog No. A15529 p110α 抑制剂MLN1117，也称为INK1117和TAK-117，是具有潜在抗肿瘤活性的I类磷酸肌醇3激酶（PI3K）α同工型的生物利用抑制剂。 了解更多
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