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搜索结果：“263”

“263”的搜索结果

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Endoxifen

Catalog No. A12639
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Estrogen receptor 拮抗剂

Endoxifen是他莫昔芬的次生代谢产物。它是负责他莫昔芬在ER阳性乳腺癌中有效性的主要代谢物。Endoxifen Z-isomer抑制hERG, 这种作用具有浓度依赖性, IC50值为1.6μM。了解更多

Product Citations (2)

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- Marina Arino Martin, .et al. Photolytic fate of (E)- and (Z)-endoxifen in water and treated wastewater exposed to sunlight, Environ Res, 2021, Apr 3;197:111121 PMID: 33823193
- Martin MA, .et al. Photodegradation of (E)- and (Z)-Endoxifen in water by ultraviolet light: Efficiency, kinetics, by-products, and toxicity assessment, Water Res, 2019, Dec 29;171:115451 PMID: 31901682
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MBX-2982

Catalog No. A12634
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GPR119 激动剂

MBX-2982是针对2型糖尿病的潜在一流疗法，其靶向G蛋白偶联受体119（GPR119），该受体与已知刺激葡萄糖依赖性胰岛素分泌的生物活性脂质相互作用。了解更多

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GSK1292263

Catalog No. A10439
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GPR119 激动剂

GSK-1292263是一种新型GPR119激动剂。了解更多

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- Inoue A, .et al. Illuminating G-Protein-Coupling Selectivity of GPCRs, Cell, 2019, Jun 13;177(7):1933-1947 PMID: 31160049