“Ligand-gated Ion Channels”的搜索结果

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  1. beta-Pompilidotoxin

    Catalog No. A15422
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    Slows neuronal Na+ channel inactivation
    beta-Pompilidotoxin是具有序列H2N-Arg的肽。 了解更多
  2. Nav1.7-IN-3

    Catalog No. A13626
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    voltage-gated sodium channel Nav1.7 inhibitor
    Nav1.7-IN-3 is a selective, orally bioavailable voltage-gated sodium channel Nav1.7 inhibitor with an IC50 of 8 nM. Pain relief. Limited CNS penetration. 了解更多
  3. Ralfinamide mesylate

    Catalog No. A22002
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    Na+ channel blocker
    Ralfinamide mesylate (FCE-26742A mesylate) is an orally available Na+ channel blocker derived from α-aminoamide, with function of suppressing pain. 了解更多
  4. Proparacaine HCl

    Catalog No. A11715
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    Voltage-gated sodium channels 拮抗剂
    Proparacaine HCl是一种电压门控钠通道拮抗剂,ED50为3.4 mM。 了解更多
  5. ICA-121431

    Catalog No. A13773
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    NaV1.3 and NaV1.1 channels 抑制剂
    ICA-121431是人NaV1.3和NaV1.1通道的有效和选择性抑制剂(IC50值分别为13和23 nM)。 了解更多
  6. Vernakalant HCl

    Catalog No. A15275
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    Ion channel blocker
    Vernakalant hydrochloride是一种研究性混合离子通道阻滞剂,可以以2至5 mg/kg的剂量终止人的急性心房纤颤(AF),并且与现有药物相比,对房颤的选择性更高。在抗心律不齐的治疗中。 了解更多

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